Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 50046761
TargetLIM domain kinase 1(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50130039(CHEMBL3629276)
Affinity DataIC50:  10nMAssay Description:Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 1(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50130038(CHEMBL3629277)
Affinity DataIC50:  11nMAssay Description:Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 1(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50130037(CHEMBL3629278)
Affinity DataIC50:  19nMAssay Description:Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 1(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50130036(CHEMBL3629279)
Affinity DataIC50:  55nMAssay Description:Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 1(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50130035(CHEMBL3629280)
Affinity DataIC50:  85nMAssay Description:Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50130036(CHEMBL3629279)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50130037(CHEMBL3629278)
Affinity DataIC50:  2.01E+3nMAssay Description:Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50130038(CHEMBL3629277)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50130035(CHEMBL3629280)
Affinity DataIC50:  4.51E+3nMAssay Description:Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50130039(CHEMBL3629276)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed