Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50046947
TargetTRAF2 and NCK-interacting protein kinase(Homo sapiens (Human))
Sree Chaitanya College

Curated by ChEMBL
LigandPNGBDBM50139421(CHEMBL3764451)
Affinity DataKi:  100nMAssay Description:Inhibition of TNIK (unknown origin) by ATP competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Sree Chaitanya College

Curated by ChEMBL
LigandPNGBDBM50139419(CHEMBL3763303)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged TRKA cytoplasmic domain (residues 440)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sree Chaitanya College

Curated by ChEMBL
LigandPNGBDBM50139420(CHEMBL3763630)
Affinity DataIC50:  33nMAssay Description:Inhibition of recombinant human CK1epsilon using GST-p53 (1 to 64 residues) as substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Sree Chaitanya College

Curated by ChEMBL
LigandPNGBDBM50025020(CHEMBL3337854)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant rat GST-tagged CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) as substrate by SDS-PAGE based autor...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Sree Chaitanya College

Curated by ChEMBL
LigandPNGBDBM50139420(CHEMBL3763630)
Affinity DataIC50:  42nMAssay Description:Inhibition of recombinant rat GST-tagged CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) as substrate by SDS-PAGE based autor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sree Chaitanya College

Curated by ChEMBL
LigandPNGBDBM50025020(CHEMBL3337854)
Affinity DataIC50:  199nMAssay Description:Inhibition of recombinant human CK1epsilon using GST-p53 (1 to 64 residues) as substrate by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sree Chaitanya College

Curated by ChEMBL
LigandPNGBDBM1894(1-(2-phenylethyl)-3-1,3-thiazol-2-ylthiourea | CHE...)
Affinity DataIC50:  900nMAssay Description:Inhibition of HIV-1 reverse transcriptase using and rCdC as template and tritium-labeled dGTP incubated for 30 mins by liquid scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed