Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50046979
TargetProstaglandin E synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50140689(CHEMBL3752809)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of PGES-1 in IL-1beta stimulated human A549 cell microsomes using PGH2 as substrate assessed as suppression of PGE2 formation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50140688(CHEMBL3754377)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of PGES-1 in IL-1beta stimulated human A549 cell microsomes using PGH2 as substrate assessed as suppression of PGE2 formation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50006805(3-(1-(4-chlorobenzyl)-3-(tert-butylthio)-5-isoprop...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of PGES-1 in IL-1beta stimulated human A549 cell microsomes using PGH2 as substrate assessed as suppression of PGE2 formation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50140689(CHEMBL3752809)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of PGES-1 in IL-1beta stimulated human A549 cell microsomes using PGH2 as substrate assessed as suppression of PGE2 formation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50140690(CHEMBL3752963)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of PGES-1 in IL-1beta stimulated human A549 cell microsomes using PGH2 as substrate assessed as suppression of PGE2 formation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50140687(CHEMBL3752388)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of PGES-1 in IL-1beta stimulated human A549 cell microsomes using PGH2 as substrate assessed as suppression of PGE2 formation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50140686(CHEMBL538661)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of PGES-1 in IL-1beta stimulated human A549 cell microsomes using PGH2 as substrate assessed as suppression of PGE2 formation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed