Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50047245
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
High Magnetic Field Laboratory

Curated by ChEMBL
LigandPNGBDBM50156123(CHEMBL3780219)
Affinity DataIC50:  62nMAssay Description:Inhibition of full length recombinant GST-tagged human p38-alpha expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
High Magnetic Field Laboratory

Curated by ChEMBL
LigandPNGBDBM50156123(CHEMBL3780219)
Affinity DataIC50:  70nMAssay Description:Inhibition of full length recombinant human ABL1 expressed in Baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
High Magnetic Field Laboratory

Curated by ChEMBL
LigandPNGBDBM50156123(CHEMBL3780219)
Affinity DataIC50:  90nMAssay Description:Inhibition of full length recombinant human C-terminal His-tagged SRC expressed in Baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
High Magnetic Field Laboratory

Curated by ChEMBL
LigandPNGBDBM50156123(CHEMBL3780219)
Affinity DataIC50:  292nMAssay Description:Inhibition of GST-tagged human DDR1 (440 to 876 residues) expressed in Baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiscoidin domain-containing receptor 2(Homo sapiens (Human))
High Magnetic Field Laboratory

Curated by ChEMBL
LigandPNGBDBM50156123(CHEMBL3780219)
Affinity DataIC50:  457nMAssay Description:Inhibition of recombinant human GST-tagged DDR2 expressed in Baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
High Magnetic Field Laboratory

Curated by ChEMBL
LigandPNGBDBM50156123(CHEMBL3780219)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of His-tagged recombinant human c-Kit without catalytic domain expressed in mammalian expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
High Magnetic Field Laboratory

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataKd:  1nMAssay Description:Binding affinity to SRC (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
High Magnetic Field Laboratory

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  27nMAssay Description:Binding affinity to P38-alpha (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
High Magnetic Field Laboratory

Curated by ChEMBL
LigandPNGBDBM50237710(4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifl...)
Affinity DataKd:  460nMAssay Description:Binding affinity to P38-alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
High Magnetic Field Laboratory

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  0.210nMAssay Description:Binding affinity to SRC (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank