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Found 7 Enz. Inhib. hit(s) with all data for entry = 50047019
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50278299(1-(6-(7-chloroquinazolin-4-yloxy)pyridin-3-yl)-3-(...)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143899(CHEMBL3759613)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143901(CHEMBL3758249)
Affinity DataIC50:  3.04E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143897(CHEMBL3758566)
Affinity DataIC50:  3.32E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143900(CHEMBL3758383)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143896(CHEMBL3758250)
Affinity DataIC50:  9.26E+4nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50143898(CHEMBL3759177)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant GST-fused SUMO E1 (unknown origin) using RanGAP1 as substrate after 2 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed