TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Modulation of gamma-secretase activity (unknown origin) assessed as amyloid-beta(1-42) production by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Modulation of gamma-secretase activity (unknown origin) assessed as amyloid-beta(1-42) production by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Modulation of gamma-secretase activity (unknown origin) assessed as amyloid-beta(1-42) production by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Modulation of gamma-secretase activity (unknown origin) assessed as amyloid-beta(1-42) production by ELISAMore data for this Ligand-Target Pair