Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50047511
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50148270(CHEMBL3739699)
Affinity DataIC50:  360nMAssay Description:Competitive binding affinity to His-tagged BRAZ2B (unknown origin) expressed in Escherichia coli BL21(DE3) cells by AlphaScreen assay in presence of ...More data for this Ligand-Target Pair
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172133(CHEMBL3809185)
Affinity DataIC50:  8.55E+3nMAssay Description:Competitive binding affinity to His-tagged BRAZ2B (unknown origin) expressed in Escherichia coli BL21(DE3) cells by AlphaScreen assay in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172116(CHEMBL3809983)
Affinity DataIC50:  2.70E+4nMAssay Description:Competitive binding affinity to His-tagged BRAZ2B (unknown origin) expressed in Escherichia coli BL21(DE3) cells by AlphaScreen assay in presence of ...More data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172111(CHEMBL3808729)
Affinity DataKd:  1.20E+4nMAssay Description:Competitive binding affinity to CBP (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172112(CHEMBL3809834)
Affinity DataKd:  6.20E+3nMAssay Description:Competitive binding affinity to CBP (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172113(CHEMBL3809636)
Affinity DataKd:  9.80E+3nMAssay Description:Competitive binding affinity to CBP (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172107(CHEMBL3810303)
Affinity DataKd:  5.30E+3nMAssay Description:Competitive binding affinity to BRD9 bromodomain (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172109(CHEMBL3809575)
Affinity DataKd:  3.50E+3nMAssay Description:Competitive binding affinity to BRD9 bromodomain (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172110(CHEMBL3809876)
Affinity DataKd:  6.30E+3nMAssay Description:Competitive binding affinity to BRD9 bromodomain (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172113(CHEMBL3809636)
Affinity DataKd: >5.00E+4nMAssay Description:Competitive binding affinity to BRD9 bromodomain (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeregrin(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172107(CHEMBL3810303)
Affinity DataKd:  1.50E+4nMAssay Description:Competitive binding affinity to human His-tagged BRPF1b (626 to 740 residues) expressed in T7 phage-infected Escherichia coli BL21(DE3) cells measure...More data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172107(CHEMBL3810303)
Affinity DataKd:  2.00E+4nMAssay Description:Competitive binding affinity to human His-tagged CREBBP (1081 to 1097 residues) expressed in T7 phage-infected Escherichia coli BL21(DE3) cells measu...More data for this Ligand-Target Pair
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM71168(2-chloranyl-N-(1-ethanoylindol-3-yl)-N-phenyl-etha...)
Affinity DataKd: >5.00E+4nMAssay Description:Competitive binding affinity to human His-tagged BRAZ2B (1858 to 1972 residues) expressed in T7 phage-infected Escherichia coli BL21(DE3) cells measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172114(CHEMBL3808440)
Affinity DataKd:  1.40E+5nMAssay Description:Competitive binding affinity to human His-tagged BRAZ2B (1858 to 1972 residues) expressed in T7 phage-infected Escherichia coli BL21(DE3) cells measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172115(CHEMBL3810055)
Affinity DataKd:  2.30E+4nMAssay Description:Competitive binding affinity to human His-tagged BRAZ2B (1858 to 1972 residues) expressed in T7 phage-infected Escherichia coli BL21(DE3) cells measu...More data for this Ligand-Target Pair
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172116(CHEMBL3809983)
Affinity DataKd:  3.90E+4nMAssay Description:Competitive binding affinity to human His-tagged BRAZ2B (1858 to 1972 residues) expressed in T7 phage-infected Escherichia coli BL21(DE3) cells measu...More data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172110(CHEMBL3809876)
Affinity DataKd:  9.30E+3nMAssay Description:Competitive binding affinity to CBP (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172109(CHEMBL3809575)
Affinity DataKd:  1.70E+4nMAssay Description:Competitive binding affinity to CBP (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172107(CHEMBL3810303)
Affinity DataKd:  2.00E+4nMAssay Description:Competitive binding affinity to CBP (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172108(CHEMBL3809158)
Affinity DataKd:  6.60E+3nMAssay Description:Competitive binding affinity to CBP (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed