Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 7213
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181101(N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...)
Affinity DataIC50:  4.18E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181097(N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...)
Affinity DataIC50:  4.72E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181098(N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  5.01E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181101(N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...)
Affinity DataIC50:  8.20E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181101(N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...)
Affinity DataIC50:  8.37E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181098(N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  9.59E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181097(N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...)
Affinity DataIC50:  1.01E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181095(N-(4-Hydroxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...)
Affinity DataIC50:  1.05E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181099(N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  1.15E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181101(N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181097(N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...)
Affinity DataIC50:  1.26E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181097(N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...)
Affinity DataIC50:  1.29E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181098(N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  1.29E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181098(N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  1.76E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181096(N-(4-fluorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  3.00E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181100(N-(4-Trifluoromethylbenzylidene)-2-(3,6-dimethyl-1...)
Affinity DataIC50:  3.59E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed