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Found 16 Enz. Inhib. hit(s) with all data for entry = 50047650
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180870(CHEMBL179861)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial membrane after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180868(CHEMBL3818299)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial membrane after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180867(CHEMBL3818586)
Affinity DataKi:  365nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial membrane after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180862(CHEMBL3819416)
Affinity DataKi:  430nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial membrane after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180869(CHEMBL3819001)
Affinity DataKi:  504nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial membrane after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180863(CHEMBL3819071)
Affinity DataKi:  783nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial membrane after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180865(CHEMBL3818951)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial membrane after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180868(CHEMBL3818299)
Affinity DataIC50:  4.30nMAssay Description:Binding affinity to MDM2 in human U87MG cells assessed as inhibition of MDM2/p53 protein interaction after 10 mins by quantitative sandwich immuno as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180869(CHEMBL3819001)
Affinity DataIC50:  9.80nMAssay Description:Binding affinity to MDM2 in human U87MG cells assessed as inhibition of MDM2/p53 protein interaction after 10 mins by quantitative sandwich immuno as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180862(CHEMBL3819416)
Affinity DataIC50:  12nMAssay Description:Binding affinity to MDM2 in human U87MG cells assessed as inhibition of MDM2/p53 protein interaction after 10 mins by quantitative sandwich immuno as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180865(CHEMBL3818951)
Affinity DataIC50:  12nMAssay Description:Binding affinity to MDM2 in human U87MG cells assessed as inhibition of MDM2/p53 protein interaction after 10 mins by quantitative sandwich immuno as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180863(CHEMBL3819071)
Affinity DataIC50:  15nMAssay Description:Binding affinity to MDM2 in human U87MG cells assessed as inhibition of MDM2/p53 protein interaction after 10 mins by quantitative sandwich immuno as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180867(CHEMBL3818586)
Affinity DataIC50:  25nMAssay Description:Binding affinity to MDM2 in human U87MG cells assessed as inhibition of MDM2/p53 protein interaction after 10 mins by quantitative sandwich immuno as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180864(CHEMBL3818934)
Affinity DataIC50:  78nMAssay Description:Binding affinity to MDM2 in human U87MG cells assessed as inhibition of MDM2/p53 protein interaction after 10 mins by quantitative sandwich immuno as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM31197(CHEMBL211045 | Nutlin-3 | med.21724, Compound 186)
Affinity DataIC50:  105nMAssay Description:Binding affinity to MDM2 in human U87MG cells assessed as inhibition of MDM2/p53 protein interaction after 10 mins by quantitative sandwich immuno as...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50180866(CHEMBL3819467)
Affinity DataIC50:  155nMAssay Description:Binding affinity to MDM2 in human U87MG cells assessed as inhibition of MDM2/p53 protein interaction after 10 mins by quantitative sandwich immuno as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed