Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50047596
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177676(CHEMBL3814041)
Affinity DataKd:  7.83E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177714(CHEMBL3813775)
Affinity DataKd:  2.68E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Mus musculus)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177678(CHEMBL3815136)
Affinity DataKd:  2.37E+5nMAssay Description:Binding affinity to TMR-linked 15N-labeled mouse Dvl-1 domain ( 247 to 341 residues) by fluorescence spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177679(CHEMBL3814761)
Affinity DataKd:  1.06E+4nMAssay Description:Binding affinity to TMR-labeled Dvl-1 PDZ domain (unknown origin) expressed in Escherichia coli by fluorescence spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177703(CHEMBL3814879)
Affinity DataKd:  3.20nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177704(CHEMBL3814273)
Affinity DataKd:  1.5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177705(CHEMBL3815146)
Affinity DataKd:  1.70nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177706(CHEMBL3814441)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177707(CHEMBL3814506)
Affinity DataKd:  3.80nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177708(CHEMBL3814619)
Affinity DataKd:  2nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177709(CHEMBL3814864)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177677(CHEMBL3814692)
Affinity DataKd:  5.80nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177714(CHEMBL3813775)
Affinity DataKd:  6.20nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177676(CHEMBL3814041)
Affinity DataKd:  2.5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177677(CHEMBL3814692)
Affinity DataKd:  1.12E+4nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177709(CHEMBL3814864)
Affinity DataKd:  6.84E+4nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177708(CHEMBL3814619)
Affinity DataKd:  3.83E+4nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177707(CHEMBL3814506)
Affinity DataKd:  1.52E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177706(CHEMBL3814441)
Affinity DataKd:  2.51E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177705(CHEMBL3815146)
Affinity DataKd:  3.11E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177704(CHEMBL3814273)
Affinity DataKd:  1.39E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177703(CHEMBL3814879)
Affinity DataKd:  6.24E+4nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177677(CHEMBL3814692)
Affinity DataKd:  186nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by fluorescence spect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed