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Found 50 Enz. Inhib. hit(s) with all data for entry = 50047422
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166849(CHEMBL3797651)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166863(CHEMBL3799529)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166852(CHEMBL3797717)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166844(CHEMBL3798478)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166859(CHEMBL3799120)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166846(CHEMBL3797435)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166861(CHEMBL3799448)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166862(CHEMBL3798490)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166853(CHEMBL3798953)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166856(CHEMBL3800251)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166860(CHEMBL3799330)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166854(CHEMBL3799638)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166847(CHEMBL3800539)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166849(CHEMBL3797651)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166850(CHEMBL3799547)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166859(CHEMBL3799120)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166843(CHEMBL3797293)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166851(CHEMBL3798840)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166862(CHEMBL3798490)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166858(CHEMBL3800153)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166848(CHEMBL3800150)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166855(CHEMBL3800576)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166847(CHEMBL3800539)
Affinity DataKi:  108nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166850(CHEMBL3799547)
Affinity DataKi:  113nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166857(CHEMBL3800055)
Affinity DataKi:  129nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166846(CHEMBL3797435)
Affinity DataKi:  205nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166842(CHEMBL3800442)
Affinity DataKi:  231nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166848(CHEMBL3800150)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166852(CHEMBL3797717)
Affinity DataKi:  367nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166844(CHEMBL3798478)
Affinity DataKi:  382nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166854(CHEMBL3799638)
Affinity DataKi:  547nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166853(CHEMBL3798953)
Affinity DataKi:  614nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166851(CHEMBL3798840)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166856(CHEMBL3800251)
Affinity DataKi:  640nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166858(CHEMBL3800153)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166863(CHEMBL3799529)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166860(CHEMBL3799330)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166861(CHEMBL3799448)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166845(CHEMBL3799430)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor in HEK293 cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166857(CHEMBL3800055)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166855(CHEMBL3800576)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166842(CHEMBL3800442)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166845(CHEMBL3799430)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166843(CHEMBL3797293)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]NMSP from human dopamine D2S receptor expressed in CHO cell membrane incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166852(CHEMBL3797717)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-benzyloxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence analysis in prese...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166863(CHEMBL3799529)
Affinity DataIC50: <1.10E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using 7-benzyloxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence analysis in prese...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166863(CHEMBL3799529)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human ERG1 expressed in CHO cells by whole cell patch clamp electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166852(CHEMBL3797717)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human ERG1 expressed in CHO cells by whole cell patch clamp electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166852(CHEMBL3797717)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human recombinant CYP2D6 using AMMC as substrate incubated for 45 mins by fluorescence analysis in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50166863(CHEMBL3799529)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CYP2D6 using AMMC as substrate incubated for 45 mins by fluorescence analysis in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed