TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 3.43E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 4.17E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 7.27E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 7.84E+3nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of N-terminal His-tagged Mer kinase (588 to 855 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells measured every mi...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Beijing Institute Of Pharmacology & Toxicology
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair