Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50047740
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50187237(CHEMBL3828515)
Affinity DataIC50:  2.81E+3nMAssay Description:Antagonist activity at RXRalpha (unknown origin) expressed in HEK293T cells assessed as inhibition of receptor transactivation after 12 hrs in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50187237(CHEMBL3828515)
Affinity DataKd:  910nMAssay Description:Binding affinity to RXRalpha-LBD (unknown origin) measured up to 300 sec by surface plasma resonance methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed