Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50047874
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50191064(CHEMBL3894220)
Affinity DataIC50:  9nMAssay Description:Antagonist activity at human P2X7 receptor assessed as reduction in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190913(CHEMBL3912682)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at human P2X7 receptor assessed as reduction in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190797(CHEMBL3974590)
Affinity DataIC50:  35nMAssay Description:Antagonist activity at human P2X7 receptor assessed as reduction in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190804(CHEMBL3966074)
Affinity DataIC50:  64nMAssay Description:Antagonist activity at human P2X7 receptor assessed as reduction in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50191067(CHEMBL3963395)
Affinity DataIC50:  78nMAssay Description:Antagonist activity at human P2X7 receptor assessed as reduction in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190797(CHEMBL3974590)
Affinity DataIC50:  80nMAssay Description:Antagonist activity at mouse P2X7 receptor assessed as reduction in calcium flux by FLIPR calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190917(CHEMBL3918589)
Affinity DataIC50:  82nMAssay Description:Antagonist activity at human P2X7 receptor assessed as reduction in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50191061(CHEMBL3893653)
Affinity DataIC50:  85nMAssay Description:Antagonist activity at human P2X7 receptor assessed as reduction in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190797(CHEMBL3974590)
Affinity DataIC50:  87nMAssay Description:Antagonist activity at P2X7 receptor in human whole blood assessed as reduction in LPS/BzATP-induced IL-1beta release preincubated with LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190913(CHEMBL3912682)
Affinity DataIC50:  103nMAssay Description:Antagonist activity at mouse P2X7 receptor assessed as reduction in calcium flux by FLIPR calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50191063(CHEMBL3982581)
Affinity DataIC50:  120nMAssay Description:Antagonist activity at human P2X7 receptor assessed as reduction in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190804(CHEMBL3966074)
Affinity DataIC50:  123nMAssay Description:Antagonist activity at mouse P2X7 receptor assessed as reduction in calcium flux by FLIPR calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190804(CHEMBL3966074)
Affinity DataIC50:  141nMAssay Description:Antagonist activity at P2X7 receptor in human whole blood assessed as reduction in LPS/BzATP-induced IL-1beta release preincubated with LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190911(CHEMBL3903665)
Affinity DataIC50:  151nMAssay Description:Antagonist activity at human P2X7 receptor assessed as reduction in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190917(CHEMBL3918589)
Affinity DataIC50:  305nMAssay Description:Antagonist activity at mouse P2X7 receptor assessed as reduction in calcium flux by FLIPR calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190797(CHEMBL3974590)
Affinity DataIC50:  316nMAssay Description:Antagonist activity at P2X7 receptor in C57/bl6 mouse whole blood assessed as reduction in LPS/BzATP-induced IL-1beta release preincubated with LPS-s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190913(CHEMBL3912682)
Affinity DataIC50:  376nMAssay Description:Antagonist activity at P2X7 receptor in human whole blood assessed as reduction in LPS/BzATP-induced IL-1beta release preincubated with LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50191061(CHEMBL3893653)
Affinity DataIC50:  486nMAssay Description:Antagonist activity at mouse P2X7 receptor assessed as reduction in calcium flux by FLIPR calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190913(CHEMBL3912682)
Affinity DataIC50:  631nMAssay Description:Antagonist activity at P2X7 receptor in C57/bl6 mouse whole blood assessed as reduction in LPS/BzATP-induced IL-1beta release preincubated with LPS-s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50190804(CHEMBL3966074)
Affinity DataIC50:  631nMAssay Description:Antagonist activity at P2X7 receptor in C57/bl6 mouse whole blood assessed as reduction in LPS/BzATP-induced IL-1beta release preincubated with LPS-s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50191064(CHEMBL3894220)
Affinity DataIC50:  1.09E+3nMAssay Description:Antagonist activity at mouse P2X7 receptor assessed as reduction in calcium flux by FLIPR calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed