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Found 24 Enz. Inhib. hit(s) with all data for entry = 50049110
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234609(Cariporide | HOE-642)
Affinity DataIC50:  172nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234607(CHEMBL4071353)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234598(CHEMBL4095965)
Affinity DataIC50:  5.09E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM32701(1-benzotriazolyl(phenyl)methanone | Benzotriazol-1...)
Affinity DataIC50:  5.16E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234612(CHEMBL4082866)
Affinity DataIC50:  5.92E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234601(CHEMBL4072374)
Affinity DataIC50:  6.06E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234602(CHEMBL557236)
Affinity DataIC50:  6.35E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234616(CHEMBL4074684)
Affinity DataIC50:  6.51E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinam...)
Affinity DataIC50:  6.67E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234604(CHEMBL425230)
Affinity DataIC50:  6.81E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234614(CHEMBL4084954)
Affinity DataIC50:  6.98E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234610(CHEMBL204234)
Affinity DataIC50:  7.24E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234596(CHEMBL1884989)
Affinity DataIC50:  7.25E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234606(CHEMBL4097403)
Affinity DataIC50:  8.65E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234617(CHEMBL3086212)
Affinity DataIC50:  9.71E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234603(CHEMBL4072288)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234615(CHEMBL4063302)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234605(CHEMBL4087253)
Affinity DataIC50:  1.35E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234600(CHEMBL4093129)
Affinity DataIC50:  1.55E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234599(CHEMBL4100842)
Affinity DataIC50:  1.57E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234608(CHEMBL4068558)
Affinity DataIC50:  1.77E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234611(CHEMBL4085368)
Affinity DataIC50:  1.91E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234613(1H-Benzo[D][1,2,3]Triazole | 1H-Benzotriazole | Be...)
Affinity DataIC50:  1.93E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 1(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234597(CHEMBL4079373)
Affinity DataIC50:  3.55E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed