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Found 192 Enz. Inhib. hit(s) with all data for entry = 50048096
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204304(CHEMBL3954961)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204312(CHEMBL3936289)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204323(CHEMBL3958393)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204321(CHEMBL3904569)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204310(CHEMBL3948140)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204320(CHEMBL3917750)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204308(CHEMBL3980626)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204300(CHEMBL3910552)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204316(CHEMBL3945203)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204305(CHEMBL3890935)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204326(CHEMBL3918997)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204307(CHEMBL3926713)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204317(CHEMBL3946273)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204298(CHEMBL3889737)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204299(CHEMBL3898676)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204322(CHEMBL3889749)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204302(CHEMBL3908975)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204297(CHEMBL3918389)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204314(CHEMBL3981067)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204309(CHEMBL3970903)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204303(CHEMBL3935644)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204325(CHEMBL3945795)
Affinity DataKi:  137nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204318(CHEMBL3959852)
Affinity DataKi:  171nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204324(CHEMBL3952259)
Affinity DataKi:  189nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204313(CHEMBL3951093)
Affinity DataKi:  209nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204305(CHEMBL3890935)
Affinity DataKi:  278nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204311(CHEMBL3907688)
Affinity DataKi:  345nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204313(CHEMBL3951093)
Affinity DataKi:  372nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204301(CHEMBL3927338)
Affinity DataKi:  407nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204306(CHEMBL3897499)
Affinity DataKi:  416nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204306(CHEMBL3897499)
Affinity DataKi:  423nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204309(CHEMBL3970903)
Affinity DataKi:  493nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204323(CHEMBL3958393)
Affinity DataKi:  632nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK cells after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204308(CHEMBL3980626)
Affinity DataKi:  638nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204312(CHEMBL3936289)
Affinity DataKi:  661nMAssay Description:Binding affinity to human M3 receptor expressed in CHO cells measured after 90 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204310(CHEMBL3948140)
Affinity DataKi:  711nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204319(CHEMBL3927917)
Affinity DataKi:  722nMAssay Description:Displacement of [3H]pentazocine from guinea pig sigma1 receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204312(CHEMBL3936289)
Affinity DataKi:  814nMAssay Description:Displacement of [3H]alpha-methylhistamine from human H3 receptor expressed in HEK Flp-In cells measured after 90 mins by microbeta scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204317(CHEMBL3946273)
Affinity DataKi:  892nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK cells after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204306(CHEMBL3897499)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]Rauwolscine from human Alpha2C receptor expressed in MDCK cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204306(CHEMBL3897499)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]Rauwolscine from human Alpha2B receptor expressed in HEK-T cells measured after 90 mins by microbeta scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204316(CHEMBL3945203)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204326(CHEMBL3918997)
Affinity DataKi:  1.28E+3nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204300(CHEMBL3910552)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204317(CHEMBL3946273)
Affinity DataKi:  1.47E+3nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204306(CHEMBL3897499)
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [3H]Rauwolscine from human Alpha2A receptor expressed in MDCK cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204322(CHEMBL3889749)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204312(CHEMBL3936289)
Affinity DataKi:  1.68E+3nMAssay Description:Displacement of [3H]Mesulergine from human 5-HT2C receptor expressed in Flp-IN HEK cells measured after 90 mins by microbeta scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50204318(CHEMBL3959852)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEKT cells measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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