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Found 12 Enz. Inhib. hit(s) with all data for entry = 7840
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM222044(5'-O-(4''-Bromobenzoyl)-thymidine-3...)
Affinity DataKi:  7.81E+3nM ΔG°:  -29.6kJ/moleT: 2°CAssay Description:In kinetic assay, the TP enzyme (0.058 U/well) was incu- bated with different concentrations of inhibitor (0.5¿0.001 mM) for 10 min at 30 C. The rea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM222045(5'-O-(3''-Bromobenzoyl)-thymidine (15))
Affinity DataKi:  1.14E+4nM ΔG°:  -28.7kJ/moleT: 2°CAssay Description:In kinetic assay, the TP enzyme (0.058 U/well) was incu- bated with different concentrations of inhibitor (0.5¿0.001 mM) for 10 min at 30 C. The rea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM222040(5'-O-(4''-Methylbenzoyl)-thymidine (4))
Affinity DataKi:  1.25E+4nM ΔG°:  -28.5kJ/moleT: 2°CAssay Description:In kinetic assay, the TP enzyme (0.058 U/well) was incu- bated with different concentrations of inhibitor (0.5¿0.001 mM) for 10 min at 30 C. The rea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM222041(5'-O-(4''-Methoxybenzoyl)-thymidine (1...)
Affinity DataKi:  1.28E+4nM ΔG°:  -28.4kJ/moleT: 2°CAssay Description:In kinetic assay, the TP enzyme (0.058 U/well) was incu- bated with different concentrations of inhibitor (0.5¿0.001 mM) for 10 min at 30 C. The rea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM50134399(1,7-Dihydro-pyrrolo[2,3-d]pyrimidine-2,4-dione | 7...)
Affinity DataKi:  4.91E+4nM ΔG°:  -25.0kJ/moleT: 2°CAssay Description:In kinetic assay, the TP enzyme (0.058 U/well) was incu- bated with different concentrations of inhibitor (0.5¿0.001 mM) for 10 min at 30 C. The rea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM222044(5'-O-(4''-Bromobenzoyl)-thymidine-3...)
Affinity DataIC50:  7.50E+3nMT: 2°CAssay Description:TP inhibition assay was performed spectrophotometrically in 96-well plate. The method of Bera et al. was followed with slight modifications [Bera et ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM222040(5'-O-(4''-Methylbenzoyl)-thymidine (4))
Affinity DataIC50:  1.85E+4nMT: 2°CAssay Description:TP inhibition assay was performed spectrophotometrically in 96-well plate. The method of Bera et al. was followed with slight modifications [Bera et ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM222041(5'-O-(4''-Methoxybenzoyl)-thymidine (1...)
Affinity DataIC50:  1.88E+4nMT: 2°CAssay Description:TP inhibition assay was performed spectrophotometrically in 96-well plate. The method of Bera et al. was followed with slight modifications [Bera et ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM222045(5'-O-(3''-Bromobenzoyl)-thymidine (15))
Affinity DataIC50:  3.33E+4nMT: 2°CAssay Description:TP inhibition assay was performed spectrophotometrically in 96-well plate. The method of Bera et al. was followed with slight modifications [Bera et ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM50134399(1,7-Dihydro-pyrrolo[2,3-d]pyrimidine-2,4-dione | 7...)
Affinity DataIC50:  4.10E+4nMT: 2°CAssay Description:TP inhibition assay was performed spectrophotometrically in 96-well plate. The method of Bera et al. was followed with slight modifications [Bera et ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM222042(5'-O-(2''-Methoxybenzoyl)-thymidine (1...)
Affinity DataIC50:  9.00E+4nMT: 2°CAssay Description:TP inhibition assay was performed spectrophotometrically in 96-well plate. The method of Bera et al. was followed with slight modifications [Bera et ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
University Of Karachi

LigandPNGBDBM222043(5'-O-(2'',4''-Dichlorobenzoyl)...)
Affinity DataIC50:  1.46E+5nMT: 2°CAssay Description:TP inhibition assay was performed spectrophotometrically in 96-well plate. The method of Bera et al. was followed with slight modifications [Bera et ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed