Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50049092
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234288(CHEMBL4085113)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234283(CHEMBL4060165)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234285(CHEMBL4083894)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234284(CHEMBL4083473)
Affinity DataKi:  3.80E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234291(CHEMBL4068819)
Affinity DataKi:  7.30E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234287(CHEMBL4100876)
Affinity DataKi:  7.70E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234280(CHEMBL4071517)
Affinity DataKi:  8.30E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234279(CHEMBL4078902)
Affinity DataKi:  1.77E+5nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234278(CHEMBL4103180)
Affinity DataKi:  1.90E+5nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234282(CHEMBL4097017)
Affinity DataKi:  1.95E+5nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234286(CHEMBL4064465)
Affinity DataKi:  2.20E+5nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234292(CHEMBL4080252)
Affinity DataKi:  3.60E+5nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234290(CHEMBL4098554)
Affinity DataKi:  3.73E+5nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Binghamton University

Curated by ChEMBL
LigandPNGBDBM50234289(CHEMBL4068036)
Affinity DataKi:  2.00E+6nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed