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Found 42 Enz. Inhib. hit(s) with all data for entry = 50049017
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232938(CHEMBL4088509)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232930(CHEMBL4067246)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232931(CHEMBL4091845)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232936(CHEMBL4071738)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232941(CHEMBL4084087)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232940(CHEMBL4071007)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232933(CHEMBL4094388)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232937(CHEMBL4086649)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232929(CHEMBL4085733)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50399157(CHEMBL2179724)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232934(CHEMBL4098746)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232935(CHEMBL4102128)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232937(CHEMBL4086649)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232935(CHEMBL4102128)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232942(CHEMBL4077875)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232939(CHEMBL4104545)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232933(CHEMBL4094388)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232944(CHEMBL4094331)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232936(CHEMBL4071738)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232928(CHEMBL4064165)
Affinity DataKi:  311nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232939(CHEMBL4104545)
Affinity DataKi:  322nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232934(CHEMBL4098746)
Affinity DataKi:  365nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232942(CHEMBL4077875)
Affinity DataKi:  467nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232944(CHEMBL4094331)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232941(CHEMBL4084087)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232930(CHEMBL4067246)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232943(CHEMBL4090242)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232931(CHEMBL4091845)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232929(CHEMBL4085733)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232938(CHEMBL4088509)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232943(CHEMBL4090242)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232940(CHEMBL4071007)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232928(CHEMBL4064165)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232938(CHEMBL4088509)
Affinity DataIC50:  21nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 EBNA cell membranes after 30 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232941(CHEMBL4084087)
Affinity DataIC50:  25nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 EBNA cell membranes after 30 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232933(CHEMBL4094388)
Affinity DataIC50:  35nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 EBNA cell membranes after 30 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232930(CHEMBL4067246)
Affinity DataIC50:  51nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 EBNA cell membranes after 30 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232936(CHEMBL4071738)
Affinity DataIC50:  55nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 EBNA cell membranes after 30 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50200170(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataIC50:  96nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 EBNA cell membranes after 30 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232937(CHEMBL4086649)
Affinity DataIC50:  296nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 EBNA cell membranes after 30 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed