Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50048135
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205807(CHEMBL3978212)
Affinity DataKi:  350nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205815(CHEMBL3907670)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205806(CHEMBL3969839)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205814(CHEMBL3898657)
Affinity DataKi:  1.28E+5nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50031467(5-HYDROXY-2-(HYDROXYMETHYL)-4H-PYRAN-4-ONE | 5-Hyd...)
Affinity DataKi:  3.50E+5nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205807(CHEMBL3978212)
Affinity DataIC50:  1.66E+4nMAssay Description:Inhibition of tyrosinase in human MNT1 cell lysate pretreated prior to addition of L-DOPA as substrate measured after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205815(CHEMBL3907670)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of tyrosinase in human MNT1 cell lysate pretreated prior to addition of L-DOPA as substrate measured after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205806(CHEMBL3969839)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of tyrosinase in human MNT1 cell lysate pretreated prior to addition of L-DOPA as substrate measured after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205807(CHEMBL3978212)
Affinity DataIC50:  8.53E+4nMAssay Description:Inhibition of tyrosinase in human MNT1 cells assessed as suppression of melanin biosynthesis measured after 96 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205806(CHEMBL3969839)
Affinity DataIC50:  1.19E+5nMAssay Description:Inhibition of tyrosinase in human MNT1 cells assessed as suppression of melanin biosynthesis measured after 96 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205815(CHEMBL3907670)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of tyrosinase in human MNT1 cells assessed as suppression of melanin biosynthesis measured after 96 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205814(CHEMBL3898657)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of tyrosinase in human MNT1 cells assessed as suppression of melanin biosynthesis measured after 96 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205814(CHEMBL3898657)
Affinity DataIC50:  1.30E+6nMAssay Description:Inhibition of tyrosinase in human MNT1 cell lysate pretreated prior to addition of L-DOPA as substrate measured after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50031467(5-HYDROXY-2-(HYDROXYMETHYL)-4H-PYRAN-4-ONE | 5-Hyd...)
Affinity DataIC50:  2.80E+6nMAssay Description:Inhibition of tyrosinase in human MNT1 cell lysate pretreated prior to addition of L-DOPA as substrate measured after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50031467(5-HYDROXY-2-(HYDROXYMETHYL)-4H-PYRAN-4-ONE | 5-Hyd...)
Affinity DataIC50:  1.50E+7nMAssay Description:Inhibition of tyrosinase in human MNT1 cells assessed as suppression of melanin biosynthesis measured after 96 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed