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Found 10 Enz. Inhib. hit(s) with all data for entry = 50048205
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50081529((S)-2-Amino-N-{(R)-1-[({(S)-2-[N'-((S)-2-amino-3-p...)
Affinity DataIC50:  0.740nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [Leu-3,4,5-3H(N)]-Substance P from NK1 receptor in rat brain homogenate measured after 60 mins by microbeta scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50208162(CHEMBL3904919)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50208162(CHEMBL3904919)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [3H]DELT2 from DOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50208161(CHEMBL3932836)
Affinity DataIC50:  4.20nMAssay Description:Displacement of [Leu-3,4,5-3H(N)]-Substance P from NK1 receptor in rat brain homogenate measured after 60 mins by microbeta scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50081523((S)-2-Amino-N-((R)-1-{[((S)-1-hydrazinocarbonyl-2-...)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [3H]DAMGO from MOR in Sprague-Dawley rat brain homogenate measured after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50208161(CHEMBL3932836)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50081529((S)-2-Amino-N-{(R)-1-[({(S)-2-[N'-((S)-2-amino-3-p...)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]DELT2 from DOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50208161(CHEMBL3932836)
Affinity DataIC50:  74nMAssay Description:Displacement of [3H]DELT2 from DOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50081523((S)-2-Amino-N-((R)-1-{[((S)-1-hydrazinocarbonyl-2-...)
Affinity DataIC50:  230nMAssay Description:Displacement of [3H]DELT2 from DOR in Sprague-Dawley rat brain homogenate measured after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed