Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50049174
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235661(CHEMBL4088796)
Affinity DataKi:  20nMAssay Description:In vitro displacement of [3H]-LY 278584 from rat cerebral cortex 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235671(CHEMBL4097212)
Affinity DataKi:  20nMAssay Description:Inhibition of endothelin-converting enzyme in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235667(CHEMBL4080688)
Affinity DataKi:  20nMAssay Description:Inhibition of endothelin-converting enzyme in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235670(CHEMBL4079988)
Affinity DataKi:  30nMAssay Description:Inhibition of VKORC1 in rat liver microsomes in presence of 0.003 to 0.2 mM vitamin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235673(CHEMBL4060572)
Affinity DataKi:  50nMAssay Description:Inhibition of VKORC1 in rat liver microsomes in presence of 0.003 to 0.2 mM vitamin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235668(CHEMBL4098946)
Affinity DataKi:  50nMAssay Description:Inhibition of neutral endopeptidase in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235672(CHEMBL4061606)
Affinity DataKi:  60nMAssay Description:Inhibition of VKORC1 in rat liver microsomes in presence of 0.003 to 0.2 mM vitamin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235674(CHEMBL4070018)
Affinity DataKi:  90nMAssay Description:Inhibition of VKORC1 in rat liver microsomes in presence of 0.003 to 0.2 mM vitamin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235664(CHEMBL4083422)
Affinity DataKi:  90nMAssay Description:Inhibition of VKORC1 in rat liver microsomes in presence of 0.003 to 0.2 mM vitamin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235665(CHEMBL4104227)
Affinity DataKi:  100nMAssay Description:Inhibition of Endothelin-converting enzyme of guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235669(CHEMBL4080910)
Affinity DataKi:  200nMAssay Description:Inhibition of VKORC1 in rat liver microsomes in presence of 0.003 to 0.2 mM vitamin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM768(4-hydroxy-3-(1-phenylpropyl)-2H-chromen-2-one | CH...)
Affinity DataKi:  200nMAssay Description:In vitro displacement of [3H]-LY 278584 from rat cerebral cortex 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235663(CHEMBL4070271)
Affinity DataKi:  260nMAssay Description:In vitro displacement of [3H]-LY 278584 from rat cerebral cortex 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235662(CHEMBL4091210)
Affinity DataKi:  3.90E+3nMAssay Description:In vitro displacement of [3H]-LY 278584 from rat cerebral cortex 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235666(CHEMBL4104918)
Affinity DataKi:  2.20E+4nMAssay Description:Inhibition of neutral endopeptidase in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed