Found 20 Enz. Inhib. hit(s) with all data for entry = 50000892 
Affinity DataKi: 44nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 223nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 331nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 356nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 586nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 869nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.99E+3nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataKi: 2.15E+3nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.37E+3nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataKi: 5.09E+3nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataKi: 1.81E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.60E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataKi: 1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataKi: 1.11E+5nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
