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Found 32 Enz. Inhib. hit(s) with all data for entry = 50001262
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274073(CHEMBL4126651)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274076(CHEMBL1384623)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274068(CHEMBL1411671)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM42435((4-methylphenyl)methyl 5-amino-2-phenyltriazole-4-...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in cell membranes after 60 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274072(CHEMBL4126042)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274071(CHEMBL4128696)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274067(CHEMBL4128108)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in cell membranes after 60 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274074(CHEMBL4127454)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274070(CHEMBL4129358)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM48290(MLS000566310 | N-(1H-benzimidazol-2-yl)benzamide |...)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from A3 receptor in human HeLa cell membranes after 180 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from A3 receptor in human HeLa cell membranes after 180 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274076(CHEMBL1384623)
Affinity DataIC50:  380nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataIC50:  410nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274068(CHEMBL1411671)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274074(CHEMBL4127454)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM42435((4-methylphenyl)methyl 5-amino-2-phenyltriazole-4-...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM48290(MLS000566310 | N-(1H-benzimidazol-2-yl)benzamide |...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274071(CHEMBL4128696)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274067(CHEMBL4128108)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274070(CHEMBL4129358)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274073(CHEMBL4126651)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274072(CHEMBL4126042)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed