Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50001749
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366289(CHEMBL4163317)
Affinity DataIC50:  2.70E+4nMAssay Description:Binding affinity to N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB domain C8Q/C67R/C84N/E99V ...More data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366279(CHEMBL4165932)
Affinity DataIC50:  3.40E+4nMAssay Description:Binding affinity to N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB domain C8Q/C67R/C84N/E99V ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366291(CHEMBL4171221)
Affinity DataIC50:  6.20E+4nMAssay Description:Binding affinity to N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB domain C8Q/C67R/C84N/E99V ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366285(CHEMBL4164855)
Affinity DataIC50:  8.00E+4nMAssay Description:Binding affinity to N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB domain C8Q/C67R/C84N/E99V ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366286(CHEMBL4169363)
Affinity DataIC50:  1.12E+5nMAssay Description:Binding affinity to N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB domain C8Q/C67R/C84N/E99V ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366282(CHEMBL4172762)
Affinity DataIC50:  1.42E+5nMAssay Description:Binding affinity to N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB domain C8Q/C67R/C84N/E99V ...More data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366281(CHEMBL4176136)
Affinity DataIC50:  1.70E+5nMAssay Description:Binding affinity to N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB domain C8Q/C67R/C84N/E99V ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366286(CHEMBL4169363)
Affinity DataKd:  2.26E+5nMAssay Description:Binding affinity to isotopically labeled and N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50260534(CHEMBL4066375)
Affinity DataKd:  1.29E+5nMAssay Description:Binding affinity to fluorescently labeled recombinant BCL6 BTB domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50239395(CHEMBL4061302)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to fluorescently labeled recombinant BCL6 BTB domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366287(CHEMBL4175189)
Affinity DataKd:  3.20E+6nMAssay Description:Binding affinity to isotopically labeled and N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB d...More data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366279(CHEMBL4165932)
Affinity DataKd:  4.05E+5nMAssay Description:Binding affinity to isotopically labeled and N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366289(CHEMBL4163317)
Affinity DataKd:  4.40E+4nMAssay Description:Binding affinity to isotopically labeled and N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB d...More data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366291(CHEMBL4171221)
Affinity DataKd:  1.53E+5nMAssay Description:Binding affinity to isotopically labeled and N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366289(CHEMBL4163317)
Affinity DataKd:  3.60E+4nMAssay Description:Binding affinity to N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB domain C8Q/C67R/C84N/E99V ...More data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366278(CHEMBL4176551)
Affinity DataKd:  2.45E+5nMAssay Description:Binding affinity to isotopically labeled and N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366285(CHEMBL4164855)
Affinity DataKd:  1.91E+5nMAssay Description:Binding affinity to isotopically labeled and N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366284(CHEMBL4168460)
Affinity DataKd:  3.00E+4nMAssay Description:Binding affinity to fluorescently labeled recombinant BCL6 BTB domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366283(CHEMBL4176318)
Affinity DataKd:  2.21E+5nMAssay Description:Binding affinity to isotopically labeled and N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366280(CHEMBL4161441)
Affinity DataKd:  2.83E+5nMAssay Description:Binding affinity to isotopically labeled and N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366282(CHEMBL4172762)
Affinity DataKd:  2.19E+5nMAssay Description:Binding affinity to isotopically labeled and N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB d...More data for this Ligand-Target Pair