Compile Data Set for Download or QSAR
maximum 50k data
Found 91 Enz. Inhib. hit(s) with all data for entry = 50035634
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50452317(CHEMBL2094085)
Affinity DataIC50:  0.520nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50452315(CHEMBL2094086)
Affinity DataIC50:  0.620nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367385(CHEMBL605863)
Affinity DataIC50:  0.860nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367375(CHEMBL604834)
Affinity DataIC50:  1nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50452316(CHEMBL2094084)
Affinity DataIC50:  1.10nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367387(CHEMBL606503)
Affinity DataIC50:  1.20nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367380(CHEMBL605449)
Affinity DataIC50:  1.5nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367383(CHEMBL604207)
Affinity DataIC50:  1.70nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367388(CHEMBL606501)
Affinity DataIC50:  2nMAssay Description:Potency against rat brain A1 adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50452322(CHEMBL2093998)
Affinity DataIC50:  2.40nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367364(CHEMBL603990)
Affinity DataIC50:  4.60nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataIC50:  10nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367374(CHEMBL606285)
Affinity DataIC50:  10nMAssay Description:Potency against rat brain adenosine A1 receptor at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50389797(CHEMBL261482)
Affinity DataIC50:  11nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367378(CHEMBL603362)
Affinity DataIC50:  11nMAssay Description:Potency against rat brain A1 adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367367(CHEMBL603358)
Affinity DataIC50:  17nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367379(CHEMBL605239)
Affinity DataIC50:  20nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50452321(CHEMBL2093997)
Affinity DataIC50:  26nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367386(CHEMBL603571)
Affinity DataIC50:  29nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50452320(CHEMBL2093996)
Affinity DataIC50:  31nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50452318(CHEMBL2093995)
Affinity DataIC50:  33nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367368(CHEMBL606290)
Affinity DataIC50:  54nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367377(CHEMBL606289)
Affinity DataIC50:  68nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367376(CHEMBL605866)
Affinity DataIC50:  70nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367384(CHEMBL606504)
Affinity DataIC50:  104nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50407975(CHEMBL519809)
Affinity DataIC50:  105nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50452314(CHEMBL2094082)
Affinity DataIC50:  105nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367369(CHEMBL605867)
Affinity DataIC50:  120nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367370(CHEMBL603359)
Affinity DataIC50:  1.40E+3nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367372(CHEMBL605029)
Affinity DataIC50:  1.70E+3nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367366(CHEMBL606288)
Affinity DataIC50:  9.60E+3nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367363(CHEMBL603573)
Affinity DataIC50:  1.00E+4nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367371(CHEMBL603360)
Affinity DataIC50:  1.30E+4nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50407975(CHEMBL519809)
Affinity DataEC50:  720nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50452322(CHEMBL2093998)
Affinity DataEC50:  980nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367375(CHEMBL604834)
Affinity DataEC50:  1.55E+3nMAssay Description:Potency against human platelet A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367368(CHEMBL606290)
Affinity DataEC50:  3.40E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367377(CHEMBL606289)
Affinity DataEC50:  5.90E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367366(CHEMBL606288)
Affinity DataEC50: >1.00E+5nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50389797(CHEMBL261482)
Affinity DataEC50:  110nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367387(CHEMBL606503)
Affinity DataEC50:  950nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367364(CHEMBL603990)
Affinity DataEC50:  4.50E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50452314(CHEMBL2094082)
Affinity DataEC50:  4.20E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367379(CHEMBL605239)
Affinity DataEC50:  6.40E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50452316(CHEMBL2094084)
Affinity DataEC50:  340nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50452317(CHEMBL2094085)
Affinity DataEC50:  820nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367380(CHEMBL605449)
Affinity DataEC50:  1.20E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367374(CHEMBL606285)
Affinity DataEC50: >1.00E+5nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367386(CHEMBL603571)
Affinity DataEC50:  420nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50452314(CHEMBL2094082)
Affinity DataEC50:  5.80E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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