Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 50007320
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50289149(GW305074X | GW5074 | US10570155, GW5074 | US113324...)
Affinity DataIC50:  71nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50289149(GW305074X | GW5074 | US10570155, GW5074 | US113324...)
Affinity DataIC50:  77nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508623(CHEMBL4568629)
Affinity DataIC50:  110nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508624(CHEMBL4443142)
Affinity DataIC50:  420nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508630(CHEMBL4579447)
Affinity DataIC50:  420nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508618(CHEMBL4465192)
Affinity DataIC50:  450nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508616(CHEMBL4453394)
Affinity DataIC50:  480nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508623(CHEMBL4568629)
Affinity DataIC50:  700nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508618(CHEMBL4465192)
Affinity DataIC50:  830nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508621(CHEMBL4567137)
Affinity DataIC50:  840nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508624(CHEMBL4443142)
Affinity DataIC50:  940nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508627(CHEMBL4466525)
Affinity DataIC50:  990nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508616(CHEMBL4453394)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508617(CHEMBL4440668)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508626(CHEMBL4440084)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508625(CHEMBL4447362)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508627(CHEMBL4466525)
Affinity DataIC50:  3.21E+3nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508621(CHEMBL4567137)
Affinity DataIC50:  3.25E+3nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508629(CHEMBL4452197)
Affinity DataIC50:  3.54E+3nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508622(CHEMBL4526774)
Affinity DataIC50:  3.66E+3nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508626(CHEMBL4440084)
Affinity DataIC50:  3.74E+3nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508619(CHEMBL4451995)
Affinity DataIC50:  4.49E+3nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508631(CHEMBL4439021)
Affinity DataIC50:  5.16E+3nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508620(CHEMBL4471372)
Affinity DataIC50:  5.32E+3nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508625(CHEMBL4447362)
Affinity DataIC50:  5.32E+3nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508632(CHEMBL4547575)
Affinity DataIC50:  6.26E+3nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508617(CHEMBL4440668)
Affinity DataIC50:  6.32E+3nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508630(CHEMBL4579447)
Affinity DataIC50:  9.42E+3nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508619(CHEMBL4451995)
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508623(CHEMBL4568629)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of wild-type BRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508622(CHEMBL4526774)
Affinity DataIC50:  1.57E+4nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508628(CHEMBL4565371)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of CRAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50508632(CHEMBL4547575)
Affinity DataIC50:  2.68E+4nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed