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Found 21 Enz. Inhib. hit(s) with all data for entry = 5386
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  5.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  5.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  9.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  35nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  42nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  351nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  1.32E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi:  2.94E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(RAT)
Aventis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM86057(CAS_62865 | Cyamemazine | NSC_62865)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed