Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50035647
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024703(6-[(2-Chloro-ethyl)-propyl-amino]-5,6,7,8-tetrahyd...)
Affinity DataIC50:  76nMAssay Description:Inhibition of purified human kidney renin, fluorometric assay using a synthetic tetradecapeptide renin substrate at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024706(6-(2-Bromo-ethylamino)-5,6,7,8-tetrahydro-naphthal...)
Affinity DataIC50:  170nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024703(6-[(2-Chloro-ethyl)-propyl-amino]-5,6,7,8-tetrahyd...)
Affinity DataIC50:  260nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024709(6-(2-Chloro-ethylamino)-5,6,7,8-tetrahydro-naphtha...)
Affinity DataIC50:  300nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024707(6-(2-Bromo-propylamino)-5,6,7,8-tetrahydro-naphtha...)
Affinity DataIC50:  300nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024706(6-(2-Bromo-ethylamino)-5,6,7,8-tetrahydro-naphthal...)
Affinity DataIC50:  420nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024704(6-[(2-Hydroxy-ethyl)-propyl-amino]-5,6,7,8-tetrahy...)
Affinity DataIC50:  420nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024707(6-(2-Bromo-propylamino)-5,6,7,8-tetrahydro-naphtha...)
Affinity DataIC50:  1.01E+3nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024702(6-[(2-Chloro-ethyl)-methyl-amino]-5,6,7,8-tetrahyd...)
Affinity DataIC50:  1.82E+3nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024708(6-[(2-Bromo-ethyl)-propyl-amino]-5,6,7,8-tetrahydr...)
Affinity DataIC50:  1.97E+3nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024704(6-[(2-Hydroxy-ethyl)-propyl-amino]-5,6,7,8-tetrahy...)
Affinity DataIC50:  2.42E+3nMAssay Description:Inhibition of purified human kidney renin, fluorometric assay using a synthetic tetradecapeptide renin substrate at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024701(6-[(2-Chloro-ethyl)-methyl-amino]-5,6,7,8-tetrahyd...)
Affinity DataIC50:  2.97E+3nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024702(6-[(2-Chloro-ethyl)-methyl-amino]-5,6,7,8-tetrahyd...)
Affinity DataIC50:  3.72E+3nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using the natural substrate partially pure angiotensinogen at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024700(6-[Bis-(2-bromo-ethyl)-amino]-5,6,7,8-tetrahydro-n...)
Affinity DataIC50:  2.20E+4nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024705(6-[(2-Chloro-ethyl)-methyl-amino]-5,6,7,8-tetrahyd...)
Affinity DataIC50:  3.22E+4nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024700(6-[Bis-(2-bromo-ethyl)-amino]-5,6,7,8-tetrahydro-n...)
Affinity DataIC50:  4.07E+4nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024709(6-(2-Chloro-ethylamino)-5,6,7,8-tetrahydro-naphtha...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using the natural substrate partially pure angiotensinogen at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024708(6-[(2-Bromo-ethyl)-propyl-amino]-5,6,7,8-tetrahydr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
Queen'S Medical Centre

Curated by ChEMBL
LigandPNGBDBM50024705(6-[(2-Chloro-ethyl)-methyl-amino]-5,6,7,8-tetrahyd...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to displace [3H]spiperone binding from anterior pituitary Dopamine receptor D2 in the presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed