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Found 47 Enz. Inhib. hit(s) with all data for entry = 5534
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50230100(4-fluoro-N-(5-(4-fluorobenzylthio)-1,3,4-thiadiazo...)
Affinity DataKi:  44nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86859(CAS_1327207 | N-(5-(4-bromobenzylthio)-1,3,4-thiad...)
Affinity DataKi:  47nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86863(CAS_4390766 | N-(5-(3-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  64nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86875(CAS_685639 | N-(5-(benzylthio)-1,3,4-thiadiazol-2-...)
Affinity DataKi:  70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86874(CAS_44454498 | N-(5-(3-chlorobenzylthio)-1,3,4-thi...)
Affinity DataKi:  73nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86857(CAS_44454939 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  83nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86868(CAS_3643794 | N-(5-(4-bromobenzylthio)-1,3,4-thiad...)
Affinity DataKi:  89nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86856(CAS_44454904 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  92nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86860(CAS_3320545 | N-(5-(4-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  104nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86856(CAS_44454904 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  165nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86867(CAS_4573026 | N-(5-(3-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  167nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86866(CAS_44454722 | N-(5-(3-chlorobenzylthio)-1,3,4-thi...)
Affinity DataKi:  169nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86870(CAS_44454776 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  170nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86864(CAS_44454803 | N-(5-(4-methoxybenzylthio)-1,3,4-th...)
Affinity DataKi:  189nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86874(CAS_44454498 | N-(5-(3-chlorobenzylthio)-1,3,4-thi...)
Affinity DataKi:  195nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86872(CAS_42805643 | N-(5-(4-methoxybenzylthio)-1,3,4-th...)
Affinity DataKi:  195nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86864(CAS_44454803 | N-(5-(4-methoxybenzylthio)-1,3,4-th...)
Affinity DataKi:  199nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86860(CAS_3320545 | N-(5-(4-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86870(CAS_44454776 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  210nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86859(CAS_1327207 | N-(5-(4-bromobenzylthio)-1,3,4-thiad...)
Affinity DataKi:  217nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86863(CAS_4390766 | N-(5-(3-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  217nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86857(CAS_44454939 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  219nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86868(CAS_3643794 | N-(5-(4-bromobenzylthio)-1,3,4-thiad...)
Affinity DataKi:  221nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86873(CAS_3448811 | N-(5-(4-bromobenzylthio)-1,3,4-thiad...)
Affinity DataKi:  225nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86862(CAS_40833444 | N-(5-(3-chlorobenzylthio)-1,3,4-thi...)
Affinity DataKi:  247nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86872(CAS_42805643 | N-(5-(4-methoxybenzylthio)-1,3,4-th...)
Affinity DataKi:  263nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86858(CAS_2192320 | N-(5-(3-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  272nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86865(CAS_44454721 | N-(5-(4-methoxybenzylthio)-1,3,4-th...)
Affinity DataKi:  272nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86871(CAS_7946867 | N-(5-(benzylthio)-1,3,4-thiadiazol-2...)
Affinity DataKi:  334nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50230100(4-fluoro-N-(5-(4-fluorobenzylthio)-1,3,4-thiadiazo...)
Affinity DataKi:  354nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86862(CAS_40833444 | N-(5-(3-chlorobenzylthio)-1,3,4-thi...)
Affinity DataKi:  369nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86871(CAS_7946867 | N-(5-(benzylthio)-1,3,4-thiadiazol-2...)
Affinity DataKi:  400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50187566(4-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzam...)
Affinity DataKi:  400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86861(CAS_2363161 | N-(5-(4-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  406nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86875(CAS_685639 | N-(5-(benzylthio)-1,3,4-thiadiazol-2-...)
Affinity DataKi:  464nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86873(CAS_3448811 | N-(5-(4-bromobenzylthio)-1,3,4-thiad...)
Affinity DataKi:  522nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86867(CAS_4573026 | N-(5-(3-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  569nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86858(CAS_2192320 | N-(5-(3-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  718nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86866(CAS_44454722 | N-(5-(3-chlorobenzylthio)-1,3,4-thi...)
Affinity DataKi:  760nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86861(CAS_2363161 | N-(5-(4-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86869(CAS_5157299 | N-(5-(benzylthio)-1,3,4-thiadiazol-2...)
Affinity DataKi:  920nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86869(CAS_5157299 | N-(5-(benzylthio)-1,3,4-thiadiazol-2...)
Affinity DataKi:  1.14E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86865(CAS_44454721 | N-(5-(4-methoxybenzylthio)-1,3,4-th...)
Affinity DataKi:  1.26E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50187565(2-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzam...)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50187578(BAS-0338868 | CHEMBL378903 | N-(5-phenethyl-1,3,4-...)
Affinity DataKi:  2.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed