Compile Data Set for Download or QSAR
maximum 50k data
Found 46 Enz. Inhib. hit(s) with all data for entry = 5629
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92292(uPa_17)
Affinity DataKi:  0.900nM ΔG°:  -51.6kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92321(uPa_43)
Affinity DataKi:  9nM ΔG°:  -45.9kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92302(uPa_26)
Affinity DataKi:  16nM ΔG°:  -44.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92313(uPa_36)
Affinity DataKi:  18nM ΔG°:  -44.2kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92316(uPa_39)
Affinity DataKi:  21nM ΔG°:  -43.8kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92304(uPa_28)
Affinity DataKi:  33nM ΔG°:  -42.7kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138662(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-a...)
Affinity DataKi:  40nM ΔG°:  -42.2kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92287(uPa_10)
Affinity DataKi:  40nM ΔG°:  -42.2kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92319(uPa_41)
Affinity DataKi:  42nM ΔG°:  -42.1kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92293(uPa_18)
Affinity DataKi:  59nM ΔG°:  -41.3kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92308(uPa_31)
Affinity DataKi:  66nM ΔG°:  -41.0kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92320(uPa_42)
Affinity DataKi:  94nM ΔG°:  -40.1kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92318(uPa_40)
Affinity DataKi:  223nM ΔG°:  -38.0kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92305(uPa_29)
Affinity DataKi:  290nM ΔG°:  -37.3kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92294(uPa_19)
Affinity DataKi:  406nM ΔG°:  -36.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50147092(8-Amino-naphthalene-2-carboxamidine | 8-amino-2-na...)
Affinity DataKi:  450nM ΔG°:  -36.2kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92289(uPa_12)
Affinity DataKi:  610nM ΔG°:  -35.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92325(uPa_8)
Affinity DataKi:  610nM ΔG°:  -35.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataKi:  628nM ΔG°:  -35.4kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50147085(7-METHOXY-8-[1-(METHYLSULFONYL)-1H-PYRAZOL-4-YL]NA...)
Affinity DataKi:  630nM ΔG°:  -35.4kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92317(uPa_4)
Affinity DataKi:  637nM ΔG°:  -35.4kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92301(uPa_25)
Affinity DataKi:  665nM ΔG°:  -35.3kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92296(uPa_20)
Affinity DataKi:  769nM ΔG°:  -34.9kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92315(uPa_38)
Affinity DataKi:  777nM ΔG°:  -34.9kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92322(uPa_44)
Affinity DataKi:  1.25E+3nM ΔG°:  -33.7kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92314(uPa_37)
Affinity DataKi:  1.49E+3nM ΔG°:  -33.3kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92309(uPa_32)
Affinity DataKi:  3.08E+3nM ΔG°:  -31.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92298(uPa_22)
Affinity DataKi:  3.57E+3nM ΔG°:  -31.1kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92288(uPa_11)
Affinity DataKi:  4.50E+3nM ΔG°:  -30.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138663(2-naphthimidamide | CHEMBL105171 | Naphthalene-2-c...)
Affinity DataKi:  5.91E+3nM ΔG°:  -29.8kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92306(uPa_3)
Affinity DataKi:  6.39E+3nM ΔG°:  -29.6kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92324(uPa_5)
Affinity DataKi:  7.28E+3nM ΔG°:  -29.3kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92297(uPa_21)
Affinity DataKi:  7.85E+3nM ΔG°:  -29.1kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92295(uPa_2)
Affinity DataKi:  8.03E+3nM ΔG°:  -29.1kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92290(uPa_14)
Affinity DataKi:  8.70E+3nM ΔG°:  -28.9kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92307(uPa_30)
Affinity DataKi: >1.00E+4nM ΔG°: >-28.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50091818(CHEMBL61743 | Isoquinolin-3-ylamine | uPa_46)
Affinity DataKi: >3.00E+4nM ΔG°: >-25.8kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92291(uPa_16)
Affinity DataKi: >4.00E+4nM ΔG°: >-25.1kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92300(uPa_24)
Affinity DataKi: >5.00E+4nM ΔG°: >-24.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92286(uPa_1)
Affinity DataKi: >5.00E+4nM ΔG°: >-24.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92303(uPa_27)
Affinity DataKi: >5.00E+4nM ΔG°: >-24.5kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92310(uPa_33)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.8kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92311(uPa_34)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.8kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92312(uPa_35)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.8kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92323(uPa_45)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.8kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM92299(uPa_23)
Affinity DataKi: >1.04E+5nM ΔG°: >-22.7kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
In DepthDetails PubMed