Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50001461
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279604(CHEMBL4163927)
Affinity DataEC50:  4.53E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279637(CHEMBL4169848)
Affinity DataEC50:  2.89E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279613(CHEMBL4176050)
Affinity DataEC50:  3.64E+3nMAssay Description:Inhibition constant against Bacillus subtilis DNA topoisomerase III (wild type).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279614(CHEMBL4170901)
Affinity DataEC50:  5.34E+3nMAssay Description:Agonist activity at human TLR8 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279615(CHEMBL4159198)
Affinity DataEC50:  4.98E+4nMAssay Description:Inhibition constant against Bacillus subtilis azp-12 DNA topoisomerase III (mutant enzyme).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279616(CHEMBL4166427)
Affinity DataEC50:  1.90E+5nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279617(CHEMBL4172654)
Affinity DataEC50:  6.67E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279618(CHEMBL3116325)
Affinity DataEC50:  1.44E+4nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279614(CHEMBL4170901)
Affinity DataEC50:  180nMAssay Description:Inhibition constant against Bacillus subtilis DNA topoisomerase III (wild type).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50240849(1-(2-methylpropyl)-1H-imidazo[4,5-c]quinolin-4-ami...)
Affinity DataEC50:  1.14E+4nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279619(CHEMBL4162974)
Affinity DataEC50:  2.21E+3nMAssay Description:Inhibition constant against Bacillus subtilis azp-12 DNA topoisomerase III (mutant enzyme).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279620(CHEMBL4162585)
Affinity DataEC50:  3.85E+3nMAssay Description:Agonist activity at human TLR8 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279621(CHEMBL4173277)
Affinity DataEC50:  2.67E+4nMAssay Description:Agonist activity at human TLR8 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279618(CHEMBL3116325)
Affinity DataEC50:  3.70E+4nMAssay Description:Inhibition constant against Bacillus subtilis azp-12 DNA topoisomerase III (mutant enzyme).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50403022(CHEMBL2216760)
Affinity DataEC50:  2.09E+4nMAssay Description:Agonist activity at human TLR8 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50241029(1-[4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c]quino...)
Affinity DataEC50:  6.13E+3nMAssay Description:Agonist activity at human TLR8 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279619(CHEMBL4162974)
Affinity DataEC50:  600nMAssay Description:Inhibition constant against Bacillus subtilis azp-12 DNA topoisomerase III (mutant enzyme).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279622(CHEMBL4174580)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279623(CHEMBL4165438)
Affinity DataEC50:  3.33E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279624(CHEMBL4161998)
Affinity DataEC50:  3.84E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279626(CHEMBL4172215)
Affinity DataEC50:  3.21E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279627(CHEMBL4160925)
Affinity DataEC50:  1.72E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279628(CHEMBL4161057)
Affinity DataEC50:  3.06E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279629(CHEMBL3116322)
Affinity DataEC50:  2.22E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279629(CHEMBL3116322)
Affinity DataEC50:  9.88E+3nMAssay Description:Agonist activity at human TLR8 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50279630(CHEMBL4164327)
Affinity DataEC50:  2.89E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50241029(1-[4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c]quino...)
Affinity DataEC50:  1.34E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50403022(CHEMBL2216760)
Affinity DataEC50:  1.69E+3nMAssay Description:Agonist activity at human TLR7 expressed in HEK cells after 8 to 12 hrs by NFkappaB/SEAP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed