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Found 19 Enz. Inhib. hit(s) with all data for entry = 50029203
LigandPNGBDBM50030727(4''-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,...)
Affinity DataIC50:  0.310nMAssay Description:In vitro binding affinity of the compound towards Angiotensin II receptor, type 1 to displace 125I[Sar,Ile] from rat brain tissue preparationMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50030727(4''-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,...)
Affinity DataIC50:  0.330nMAssay Description:In vitro binding affinity of the compound towards Angiotensin II receptor, type 1 to displace 125I[Sar,Ile] from rat adrenal tissue preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50030727(4''-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,...)
Affinity DataIC50:  0.430nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50030727(4''-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,...)
Affinity DataIC50:  0.5nMAssay Description:In vitro binding affinity of the compound towards angiotensin-1 receptor to displace 125I[Sar,Ile] from rabbit adrenal tissue preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50030727(4''-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,...)
Affinity DataIC50:  0.550nMAssay Description:In vitro binding affinity of the compound towards angiotensin-1 receptor to displace 125I[Sar,Ile] from rabbit brain tissue preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50030727(4''-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,...)
Affinity DataIC50:  0.550nMAssay Description:In vitro binding affinity of the compound towards angiotensin-1 receptor to displace 125I[Sar,Ile] from rabbit brain tissue preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50035431(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  0.780nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282212(4'-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5...)
Affinity DataIC50:  0.800nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282213(4'-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5...)
Affinity DataIC50:  0.800nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50039888(4'-[3-Butyl-1-(2-chloro-phenyl)-5-oxo-1,5-dihydro-...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50039872(4'-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5...)
Affinity DataIC50:  1.60nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50044503(5-Butyl-2-(2,2-dimethyl-propyl)-4-[2'-(2H-tetrazol...)
Affinity DataIC50:  2.10nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50044505(5-Butyl-2-(2-chloro-phenyl)-4-[2'-(2H-tetrazol-5-y...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50039919(4'-[3-Butyl-1-(2,6-dichloro-phenyl)-5-oxo-1,5-dihy...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50039915(4'-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5...)
Affinity DataIC50:  2.90nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50039925(4''-[3-Butyl-1-(2,2-dimethyl-propyl)-5-oxo-1,5-dih...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50044479(5-Butyl-2-(2,6-dichloro-phenyl)-4-[2'-(2H-tetrazol...)
Affinity DataIC50:  5.80nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50030727(4''-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,...)
Affinity DataIC50:  270nMAssay Description:In vitro binding affinity of the compound towards Angiotensin II receptor, type 2 to displace 125I[Sar,Ile] from rat adrenal tissue preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50030727(4''-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,...)
Affinity DataIC50:  300nMAssay Description:In vitro binding affinity of the compound towards Angiotensin II receptor, type 2 to displace 125I[Sar,Ile] from rat brain tissue preparationMore data for this Ligand-Target Pair
In DepthDetails Article