Compile Data Set for Download or QSAR
maximum 50k data
Found 46 Enz. Inhib. hit(s) with all data for entry = 50029286
LigandPNGBDBM50031491(2-propyl-4-(methythio)-1-[[[2'-[(propylamino)carbo...)
Affinity DataIC50:  0.300nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283002(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50:  0.600nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283000(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50032362(3-(2'-Isopentyloxycarbonylsulfamoyl-3-fluoro-biphe...)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50032364(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50032362(3-(2'-Isopentyloxycarbonylsulfamoyl-3-fluoro-biphe...)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283000(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283001(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283006(3-(2'-Butyloxycarbonylsulfamoyl-biphenyl-4-ylmethy...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283008(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM36645(CHEMBL291582 | L-707,581)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283003(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283005(3-(2'-Butyloxycarbonylsulfamoyl-3-bromo-biphenyl-4...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50049179(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50032364(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM82428(CAS_124750-95-4 | CB91356279 | CHEMBL443269 | DuP ...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50032351(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283009(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283007(3-(2'-Butyloxycarbonylsulfamoyl-3-methyl-biphenyl-...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50049196(3-[3-Bromo-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283002(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282999(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283012(3-(2'-Butyloxycarbonylsulfamoyl-3-nitro-biphenyl-4...)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50032351(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283004(5-Ethyl-3-[3-fluoro-2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283009(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  9nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283001(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283013(3-[3-Chloro-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283007(3-(2'-Butyloxycarbonylsulfamoyl-3-methyl-biphenyl-...)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282999(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283005(3-(2'-Butyloxycarbonylsulfamoyl-3-bromo-biphenyl-4...)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283012(3-(2'-Butyloxycarbonylsulfamoyl-3-nitro-biphenyl-4...)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283010(3-[3-Bromo-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283003(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283006(3-(2'-Butyloxycarbonylsulfamoyl-biphenyl-4-ylmethy...)
Affinity DataIC50:  40nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283011(5-Ethyl-3-[3-methyl-2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  40nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50049196(3-[3-Bromo-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  80nMAssay Description:Compound was tested for the inhibition of angiotensin II AT2 receptor by displacement of [125I]- Ang II to rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283008(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  80nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283013(3-[3-Chloro-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50:  500nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50049179(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  500nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283010(3-[3-Bromo-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  700nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50031491(2-propyl-4-(methythio)-1-[[[2'-[(propylamino)carbo...)
Affinity DataIC50:  775nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283011(5-Ethyl-3-[3-methyl-2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283004(5-Ethyl-3-[3-fluoro-2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  3.00E+3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM36645(CHEMBL291582 | L-707,581)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM82428(CAS_124750-95-4 | CB91356279 | CHEMBL443269 | DuP ...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article