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Found 22 Enz. Inhib. hit(s) with all data for entry = 50029336
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  8.5nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  130nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283517(10-(3-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50:  200nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  430nMAssay Description:Binding to delta opioid receptor by using [3H]-DPDPE as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283522(4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapentacycl...)
Affinity DataIC50:  530nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283516(1-[14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-...)
Affinity DataIC50:  640nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283517(10-(3-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50:  910nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283521(10-(2-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50:  2.60E+3nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283519(4-methyl-10-(3-thienyl)-(1S,5R,13R,14S,17R)-12-oxa...)
Affinity DataIC50:  3.30E+3nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283523(4,10-dimethyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapent...)
Affinity DataIC50:  4.50E+3nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283516(1-[14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-...)
Affinity DataIC50:  5.10E+3nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283518(14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-a...)
Affinity DataIC50:  6.40E+3nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283517(10-(3-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50:  7.40E+3nMAssay Description:Binding to delta opioid receptor by using [3H]-DPDPE as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283516(1-[14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-...)
Affinity DataIC50:  7.90E+3nMAssay Description:Binding to delta opioid receptor by using [3H]-DPDPE as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283521(10-(2-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50:  9.50E+3nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283522(4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapentacycl...)
Affinity DataIC50:  1.10E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283519(4-methyl-10-(3-thienyl)-(1S,5R,13R,14S,17R)-12-oxa...)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283525(4-methyl-10-(2-thienyl)-(1S,5R,13R,14S,17R)-12-oxa...)
Affinity DataIC50:  2.50E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283523(4,10-dimethyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapent...)
Affinity DataIC50:  3.60E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283524(4-methyl-10-phenyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataIC50:  7.60E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283518(14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-a...)
Affinity DataIC50:  1.11E+5nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283520(10-benzo[b]thiophen-2-yl-4-methyl-(1S,5R,13R,14S,1...)
Affinity DataIC50:  1.26E+5nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article