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Found 32 Enz. Inhib. hit(s) with all data for entry = 50029416
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284276(CHEMBL264220 | Endothelin-1 analogue)
Affinity DataIC50:  5.27E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284276(CHEMBL264220 | Endothelin-1 analogue)
Affinity DataIC50:  5.59E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284288(CHEMBL439090 | Endothelin-1 analogue)
Affinity DataIC50:  5.77E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284286(CHEMBL411371 | Endothelin-1 analogue)
Affinity DataIC50:  6.07E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284278(CHEMBL383109 | Endothelin-1 analogue)
Affinity DataIC50:  6.13E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284284(CHEMBL216868 | Endothelin-1 analogue)
Affinity DataIC50:  6.71E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284285(CHEMBL440254 | Endothelin-1 analogue)
Affinity DataIC50:  6.85E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284281(CHEMBL383113 | Endothelin-1 analogue)
Affinity DataIC50:  7.04E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284287(CHEMBL438213 | Endothelin-1 analogue)
Affinity DataIC50:  7.53E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284278(CHEMBL383109 | Endothelin-1 analogue)
Affinity DataIC50:  7.55E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284277(CHEMBL411933 | Endothelin-1 analogue)
Affinity DataIC50:  7.59E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284289(CHEMBL382683 | Endothelin-1 analogue)
Affinity DataIC50:  7.60E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284288(CHEMBL439090 | Endothelin-1 analogue)
Affinity DataIC50:  7.96E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284279(CHEMBL439471 | Endothelin-1 analogue)
Affinity DataIC50:  7.97E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284275(CHEMBL414596 | Endothelin-1 analogue)
Affinity DataIC50:  8.06E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284285(CHEMBL440254 | Endothelin-1 analogue)
Affinity DataIC50:  8.60E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284286(CHEMBL411371 | Endothelin-1 analogue)
Affinity DataIC50:  8.60E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284283(CHEMBL439489 | Endothelin-1 analogue)
Affinity DataIC50:  8.89E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284280(CHEMBL411360 | Endothelin-1 analogue)
Affinity DataIC50:  9.00E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284280(CHEMBL411360 | Endothelin-1 analogue)
Affinity DataIC50:  9.05E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284287(CHEMBL438213 | Endothelin-1 analogue)
Affinity DataIC50:  9.40E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284277(CHEMBL411933 | Endothelin-1 analogue)
Affinity DataIC50:  9.40E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284281(CHEMBL383113 | Endothelin-1 analogue)
Affinity DataIC50:  9.59E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284283(CHEMBL439489 | Endothelin-1 analogue)
Affinity DataIC50:  9.76E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284284(CHEMBL216868 | Endothelin-1 analogue)
Affinity DataIC50:  9.77E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284275(CHEMBL414596 | Endothelin-1 analogue)
Affinity DataIC50:  9.78E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284282(CHEMBL411290 | Endothelin-1 analogue)
Affinity DataIC50:  9.88E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284290(CHEMBL412233 | Endothelin-1 analogue)
Affinity DataIC50:  9.93E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284279(CHEMBL439471 | Endothelin-1 analogue)
Affinity DataIC50:  9.94E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284282(CHEMBL411290 | Endothelin-1 analogue)
Affinity DataIC50:  1.00E+7nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284289(CHEMBL382683 | Endothelin-1 analogue)
Affinity DataIC50:  1.00E+7nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284290(CHEMBL412233 | Endothelin-1 analogue)
Affinity DataIC50:  1.01E+7nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article