Compile Data Set for Download or QSAR
maximum 50k data
Found 29 Enz. Inhib. hit(s) with all data for entry = 50029692
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataIC50:  0.110nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286903(1-[1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pyridin-2...)
Affinity DataIC50:  0.120nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286897(1-[2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-pyridin-2-yl-...)
Affinity DataIC50:  0.130nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286882(1-[(S)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50:  0.230nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50056096(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50:  0.440nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50056097(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50:  0.520nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286896(1-(3,3-Dimethyl-2-oxo-butyl)-5-thiazol-2-yl-3-[(m-...)
Affinity DataIC50:  0.800nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286904(1-[1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyrazin-2-...)
Affinity DataIC50:  0.880nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286900(1-[1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pyridin-3...)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286898(1-[1-(3,3-Dimethyl-2-oxo-butyl)-5-(1-methyl-1H-imi...)
Affinity DataIC50:  4.5nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286899(1-[1-(3,3-Dimethyl-2-oxo-butyl)-5-(1H-imidazol-2-y...)
Affinity DataIC50:  8nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286894(1-[2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-pyridin-4-yl-...)
Affinity DataIC50:  18nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286901(1-[1-(3,3-Dimethyl-2-oxo-butyl)-5-(1H-imidazol-4-y...)
Affinity DataIC50:  26nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286902(1-[1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pyridin-4...)
Affinity DataIC50:  48nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286900(1-[1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pyridin-3...)
Affinity DataIC50:  80nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50286895(1-(3,3-Dimethyl-2-oxo-butyl)-5-(1H-pyrazol-3-yl)-3...)
Affinity DataIC50: >100nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286895(1-(3,3-Dimethyl-2-oxo-butyl)-5-(1H-pyrazol-3-yl)-3...)
Affinity DataIC50:  105nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50056097(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50:  111nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataIC50:  146nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286901(1-[1-(3,3-Dimethyl-2-oxo-butyl)-5-(1H-imidazol-4-y...)
Affinity DataIC50:  232nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286896(1-(3,3-Dimethyl-2-oxo-butyl)-5-thiazol-2-yl-3-[(m-...)
Affinity DataIC50:  433nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50056096(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50:  470nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286894(1-[2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-pyridin-4-yl-...)
Affinity DataIC50:  670nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286898(1-[1-(3,3-Dimethyl-2-oxo-butyl)-5-(1-methyl-1H-imi...)
Affinity DataIC50:  844nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286897(1-[2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-pyridin-2-yl-...)
Affinity DataIC50:  980nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286904(1-[1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyrazin-2-...)
Affinity DataIC50:  1.36E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286903(1-[1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pyridin-2...)
Affinity DataIC50:  2.60E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286899(1-[1-(3,3-Dimethyl-2-oxo-butyl)-5-(1H-imidazol-2-y...)
Affinity DataIC50:  2.62E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286902(1-[1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pyridin-4...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor from rat pancreas using [I125]-L-364,718 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article