Compile Data Set for Download or QSAR
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Found 14 Enz. Inhib. hit(s) with all data for entry = 50030045
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290547((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-meth...)
Affinity DataIC50:  5.20E+3nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290549((R)-[2-(4-Chloro-phenyl)-6-methoxy-quinolin-4-yl]-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290549((R)-[2-(4-Chloro-phenyl)-6-methoxy-quinolin-4-yl]-...)
Affinity DataIC50:  5.90E+3nMAssay Description:Compound was tested in vitro for its binding affinity towards recombinant human Calcitonin gene-related peptide type receptor (membranes of HEK-293 c...More data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290551((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-meth...)
Affinity DataIC50:  9.90E+3nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290558((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-meth...)
Affinity DataIC50:  1.20E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290553((R)-[2-(3-Chloro-4-fluoro-phenyl)-6-methoxy-quinol...)
Affinity DataIC50:  1.70E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290548((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-(6-meth...)
Affinity DataIC50:  3.30E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290556((R)-[2-(2,4-Dichloro-phenyl)-6-methoxy-quinolin-4-...)
Affinity DataIC50:  3.70E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290552((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-meth...)
Affinity DataIC50:  4.10E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290550((R)-(2-Benzo[1,3]dioxol-5-yl-6-methoxy-quinolin-4-...)
Affinity DataIC50:  7.40E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290546((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-(6-meth...)
Affinity DataIC50:  9.60E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290555((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290557((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-(6-meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290554((R)-[2-(3-Amino-phenyl)-6-methoxy-quinolin-4-yl]-(...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article