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Found 20 Enz. Inhib. hit(s) with all data for entry = 50044713
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026881(CHEMBL3335530)
Affinity DataIC50:  8.00E+3nMAssay Description:Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50027066(CHEMBL3335534)
Affinity DataIC50:  8.00E+3nMAssay Description:Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026887(CHEMBL3335533)
Affinity DataIC50:  1.60E+4nMAssay Description:Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026870(CHEMBL3335528)
Affinity DataIC50:  1.80E+4nMAssay Description:Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50400720(CHEMBL2204272)
Affinity DataIC50:  1.80E+4nMAssay Description:Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026882(CHEMBL3335531)
Affinity DataIC50:  1.90E+4nMAssay Description:Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026886(CHEMBL3335532)
Affinity DataIC50:  2.10E+4nMAssay Description:Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026871(CHEMBL3335529)
Affinity DataIC50:  3.40E+4nMAssay Description:Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026881(CHEMBL3335530)
Affinity DataIC50:  6.70E+4nMAssay Description:Antagonist activity at P-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026881(CHEMBL3335530)
Affinity DataIC50:  7.60E+4nMAssay Description:Antagonist activity at E-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026870(CHEMBL3335528)
Affinity DataIC50:  1.10E+5nMAssay Description:Antagonist activity at P-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026870(CHEMBL3335528)
Affinity DataIC50:  1.40E+5nMAssay Description:Antagonist activity at E-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026871(CHEMBL3335529)
Affinity DataIC50:  1.90E+5nMAssay Description:Antagonist activity at P-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026871(CHEMBL3335529)
Affinity DataIC50:  2.20E+5nMAssay Description:Antagonist activity at E-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026869(CHEMBL3335527)
Affinity DataIC50:  5.20E+5nMAssay Description:Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50400721(CHEMBL2204273)
Affinity DataIC50:  8.80E+5nMAssay Description:Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026869(CHEMBL3335527)
Affinity DataIC50:  1.90E+6nMAssay Description:Antagonist activity at P-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50026869(CHEMBL3335527)
Affinity DataIC50:  2.08E+6nMAssay Description:Antagonist activity at E-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50400721(CHEMBL2204273)
Affinity DataIC50:  4.84E+6nMAssay Description:Antagonist activity at P-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Institut De Recherches Cliniques De Montr£Al (Ircm)

Curated by ChEMBL
LigandPNGBDBM50400721(CHEMBL2204273)
Affinity DataIC50:  5.46E+6nMAssay Description:Antagonist activity at E-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed