Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50046570
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataKi:  5.90E+4nMAssay Description:Inhibition of human recombinant serine racemase expressed in Escherichia coli Rosetta 2 (DE3) cells using L-serine as substrate by horseradish peroxi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataKi:  6.60E+4nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119563(CHEBI:45969 | TRICARBALLYLIC ACID)
Affinity DataKi:  1.30E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119565(CHEMBL3617722)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119562(CHEMBL3617724)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119564(CHEMBL3617723)
Affinity DataKi:  1.70E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119560(CHEMBL3617727)
Affinity DataKi:  4.50E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119561(CHEMBL3617725)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed