Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
GlcB (Homo sapiens (Human)) | BDBM50083940![]() (4-(3-Chloro-phenyl)-2-hydroxy-4-oxo-but-2-enoic ac...) | PDB GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM50174491![]() ((Z)-2-Hydroxy-4-oxo-4-m-tolyl-but-2-enoic acid | C...) | PDB GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM50152579![]() (4-(2-Fluoro-phenyl)-2,4-dioxo-butyric acid | CHEMB...) | PDB GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM50152554![]() (4-(2-Chloro-phenyl)-2,4-dioxo-butyric acid | CHEMB...) | PDB GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225389![]() (Sacchettini_4) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | PDB | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
GlcB (Homo sapiens (Human)) | BDBM50083953![]() ((Z)-4-(3-Bromo-phenyl)-2-hydroxy-4-oxo-but-2-enoic...) | PDB GoogleScholar AffyNet ![]() | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | PDB | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
GlcB (Homo sapiens (Human)) | BDBM50152575![]() (2,4-Dioxo-4-o-tolyl-butyric acid | CHEMBL1829214 |...) | PDB GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid PDB UniChem Patents Similars | PDB | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
GlcB (Homo sapiens (Human)) | BDBM50115579![]() ((Z)-2-hydroxy-4-oxo-4-phenyl-but-2-enoic acid | 2-...) | PDB GoogleScholar AffyNet ![]() | Purchase CHEMBL MMDB PC cid PC sid PDB UniChem Patents Similars | PDB | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225391![]() (Sacchettini_10) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225392![]() (Sacchettini_11) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | PDB | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225390![]() (Sacchettini_9) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | 5.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM50137853![]() (2,4-Dioxo-4-p-tolyl-butyric acid | 2,4-dioxo-4-p-t...) | PDB GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225399![]() (Sacchettini_26) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225394![]() (Sacchettini_21) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225398![]() (Sacchettini_25) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225393![]() (Sacchettini_20) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225396![]() (Sacchettini_23) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225397![]() (Sacchettini_24) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GlcB (Homo sapiens (Human)) | BDBM225395![]() (Sacchettini_22) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
D3R | Assay Description DNTB-Coupled_Enzyme_Assay | D3R 223: (2015) BindingDB Entry DOI: 10.7270/Q2NC602G | |||||||||||
More data for this Ligand-Target Pair |