Compile Data Set for Download or QSAR
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Found 48 Enz. Inhib. hit(s) with all data for entry = 4805
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(MOUSE)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  1.83nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
Affinity DataKi:  1.94nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  2.15nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  2.34nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  2.69nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-arrestin-1(RABBIT)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  3.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(MOUSE)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  4.80nMMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  5.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  7.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  8.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  9.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  12.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
Affinity DataKi:  13.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  13.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  14.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  15.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  16.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  18.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  18.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-arrestin-1(RABBIT)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  24nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(MOUSE)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  26nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  27.5nMMore data for this Ligand-Target Pair
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  29.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
Affinity DataKi:  35.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  37.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
Affinity DataKi:  38.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
Affinity DataKi:  39.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  58.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  58.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  63nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-arrestin-1(RABBIT)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  67.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  73nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  85nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(GUINEA PIG)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  86.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(MOUSE)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
Affinity DataKi:  127nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(MOUSE)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  159nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(MOUSE)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  320nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-arrestin-1(RABBIT)
Stanford University

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  358nMMore data for this Ligand-Target Pair
In DepthDetails PubMed