Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50004873
TargetTumor necrosis factor receptor superfamily member 16(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50029495(7-Benzoylamino-4-methyl-9-oxo-4,9-dihydro-pyrazolo...)
Affinity DataIC50:  200nMAssay Description:Inhibition of [125I]- NGF binding to extracellular domain of p75 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor receptor superfamily member 16(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50029497(2-Methyl-7-oxo-5-(tetrazol-1-ylcarbamoyl)-4,7-dihy...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of [125I]- NGF binding to extracellular domain of p75 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor receptor superfamily member 16(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50029494(2-Methyl-7-oxo-4,7-dihydro-thieno[3,2-b]pyridine-3...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of [125I]- NGF binding to extracellular domain of p75 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor necrosis factor receptor superfamily member 16(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50029496(6-Amino-4-oxo-1,4-dihydro-quinoline-2-carboxylic a...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of [125I]- NGF binding to extracellular domain of p75 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed