Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50036234
TargetMu-type opioid receptor(CALF)
Institute

Curated by ChEMBL
LigandPNGBDBM50030143(CHEMBL41098 | bis-(1N-[10-hydroxy-4-methyl-14-oxo-...)
Affinity DataIC50:  0.400nMAssay Description:Evaluation for the inhibition of mu opioid binding to bovine striatal membranes by the affinity ligand 0.25 nM [3H]DAMGO radiolabeled opioidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
Institute

Curated by ChEMBL
LigandPNGBDBM50030144(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacy...)
Affinity DataIC50:  0.630nMAssay Description:Evaluation for the inhibition of mu opioid binding to bovine striatal membranes by the affinity ligand 0.25 nM [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
Institute

Curated by ChEMBL
LigandPNGBDBM50030145(CHEMBL290701 | bis-(1N-[4-cyclopropylmethyl-10-hyd...)
Affinity DataIC50:  3.30nMAssay Description:Evaluation for the inhibition of mu opioid binding to bovine striatal membranes by the affinity ligand 0.25 nM [3H]DAMGO radiolabeled opioidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50030145(CHEMBL290701 | bis-(1N-[4-cyclopropylmethyl-10-hyd...)
Affinity DataIC50:  10nMAssay Description:Evaluation for the inhibition of kappa opioid binding to bovine striatal membranes by the affinity ligand 1 nM [3H]U-69593 radiolabeled opioidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50030143(CHEMBL41098 | bis-(1N-[10-hydroxy-4-methyl-14-oxo-...)
Affinity DataIC50:  11nMAssay Description:Evaluation for the inhibition of delta opioid binding to bovine striatal membranes by the affinity ligand 0.2 nM [3H]-p-Cl-DPDPE radiolabeled opioidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50030144(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacy...)
Affinity DataIC50:  12nMAssay Description:Evaluation for the inhibition of delta opioid binding to bovine striatal membranes by the affinity ligand 0.2 nM [3H]p-Cl-DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50030145(CHEMBL290701 | bis-(1N-[4-cyclopropylmethyl-10-hyd...)
Affinity DataIC50:  24nMAssay Description:Evaluation for the inhibition of delta opioid binding to bovine striatal membranes by the affinity ligand 0.2 nM [3H]-p-Cl-DPDPE radiolabeled opioidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50030143(CHEMBL41098 | bis-(1N-[10-hydroxy-4-methyl-14-oxo-...)
Affinity DataIC50:  41nMAssay Description:Evaluation for the inhibition of kappa opioid binding to bovine striatal membranes by the affinity ligand 1 nM [3H]-U-69,593 radiolabeled opioidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50030144(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacy...)
Affinity DataIC50:  41nMAssay Description:Evaluation for the inhibition of kappa opioid binding to bovine striatal membranes by the affinity ligand 1 nM [3H]U-69593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed