TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 0.670nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 1.72nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 1.75nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 2.49nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 2.62nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Binding affinity of the compound was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 35.2nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 35.2nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 68.6nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 70.6nMAssay Description:Binding affinity of the compound was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 71.5nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 83.1nMAssay Description:Binding affinity of the compound was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 144nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 144nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 211nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 231nMAssay Description:Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 283nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 346nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 365nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 365nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 597nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 764nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.22E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.54E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.71E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.01E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.17E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.96E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 2 using [3H]- DTG as radioligandMore data for this Ligand-Target Pair