Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50036355
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033211(7,8-Dichloro-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  0.5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033212(7,8-Dichloro-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  0.5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033213(7,8-Dichloro-1-methyl-4-[4-(2-methyl-imidazo[4,5-c...)
Affinity DataIC50:  0.5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033223(7,8-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  0.600nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033214(7,8-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  0.700nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033206(7,8-Dichloro-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  0.900nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033207(7,8-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  1.90nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033217(7,8-Dichloro-2-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  4nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004633((S)-4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-im...)
Affinity DataIC50:  4.30nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033218(1-Methyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  4.90nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033224(4-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033215(2-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  15nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033219(2-Methyl-1-[4-(5-phenyl-[1,3,4]oxadiazol-2-yl)-phe...)
Affinity DataIC50:  44nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033226(1-(4-Iodo-phenyl)-2-methyl-1H-imidazo[4,5-c]pyridi...)
Affinity DataIC50:  67nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50038755(6-(2-chlorophenyl)-1-methyl-8,9-dihydro-4H,7H-cycl...)
Affinity DataIC50:  73nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033221(5-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  190nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033225(4-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  200nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033209(1-[4-(1H-Benzoimidazol-2-yl)-phenyl]-2-methyl-1H-i...)
Affinity DataIC50:  350nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033216(3-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  600nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033208(2-Methyl-1-phenyl-1H-imidazo[4,5-c]pyridine | CHEM...)
Affinity DataIC50:  840nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033222(7-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  2.60E+3nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033220(5-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed