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Found 34 Enz. Inhib. hit(s) with all data for entry = 50005518
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM591((2R,4S)-2-[(R)-(benzylcarbamoyl)(1-phenylacetamido...)
Affinity DataIC50:  0.900nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM636((2R,4S)-2-[(R)-(benzylcarbamoyl)(1-phenylacetamido...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037825(1N-ethyl-2-benzylcarboxamido-2-[4-{2-[2-benzylcarb...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM519((2S)-N-[(2S,3R)-4-[(3S,4aS,8aS)-3-(tert-butylcarba...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037842(4N-(tert-butyl)-3-{3-[2-benzylcarbamoyl(benzylcarb...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037817((3S,4aS,8aS)-2-[(S)-3-({(2R,4S)-2-[Benzylcarbamoyl...)
Affinity DataIC50:  23nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037832((3S,4aS,8aS)-2-[(S)-3-({(2R,4S)-2-[Carbamoyl-((S)-...)
Affinity DataIC50:  23nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037833((3S,4aS,8aS)-2-[(S)-3-({(2R,4S)-2-[(4-Dimethylamin...)
Affinity DataIC50:  26nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037819((3S,4aS,8aS)-2-[3-({(2R,4S)-2-[Ethylcarbamoyl-((S)...)
Affinity DataIC50:  31nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037824(CHEMBL122641 | {(2R,4S)-4-[(S)-3-((3S,4aS,8aS)-3-t...)
Affinity DataIC50:  54nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50407257(CHEMBL2112601)
Affinity DataIC50:  58nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50407258(CHEMBL2111802)
Affinity DataIC50:  82nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037828((3S,4aS,8aS)-2-[3-({(2R,4S)-2-[Heptylcarbamoyl-((S...)
Affinity DataIC50:  86nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037835(3-[(R)-3-({(2R,4S)-2-[Benzylcarbamoyl-((S)-phenyla...)
Affinity DataIC50:  93nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037818(2-(3-{[5,5-Dimethyl-2-({2-[5-(2-oxo-hexahydro-thie...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037827(CHEMBL125827 | {2-[2-{(2R,4S)-4-[3-((3S,4aS,8aS)-3...)
Affinity DataIC50:  160nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037841((3S,4aS,8aS)-2-[(R)-3-({(2R,4S)-2-[Benzylcarbamoyl...)
Affinity DataIC50:  160nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037822(3-[(S)-3-({(2R,4S)-2-[Benzylcarbamoyl-((S)-phenyla...)
Affinity DataIC50:  190nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037834((3S,4aS,8aS)-2-[(R)-3-({(2R,4S)-2-[(Cyclohexylmeth...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037830((2R,4S)-2-[Benzylcarbamoyl-((S)-phenylacetylamino)...)
Affinity DataIC50:  450nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM635((2R,4S)-2-[(R)-(benzylcarbamoyl)(1-phenylacetamido...)
Affinity DataIC50:  540nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037836((2R,4S)-2-[Benzylcarbamoyl-((S)-phenylacetylamino)...)
Affinity DataIC50:  650nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037839((2R,4S)-2-[Ethylcarbamoyl-((S)-phenylacetylamino)-...)
Affinity DataIC50:  710nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037821((2R,4S)-2-[Ethylcarbamoyl-((S)-phenylacetylamino)-...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037829((2R,4S)-2-[Benzylcarbamoyl-((S)-phenylacetylamino)...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037826((2R,4S)-2-[Benzylcarbamoyl-((S)-phenylacetylamino)...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037840((S)-1-[(R)-3-({(2R,4S)-2-[Benzylcarbamoyl-((S)-phe...)
Affinity DataIC50: >2.20E+3nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037829((2R,4S)-2-[Benzylcarbamoyl-((S)-phenylacetylamino)...)
Affinity DataIC50:  3.10E+3nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037831((2R,4S)-2-[Benzylcarbamoyl-((S)-phenylacetylamino)...)
Affinity DataIC50:  4.60E+3nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037837((2R,4S)-2-[Benzylcarbamoyl-((S)-phenylacetylamino)...)
Affinity DataIC50:  5.10E+3nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037820((2R,4S)-2-[Benzylcarbamoyl-((S)-phenylacetylamino)...)
Affinity DataIC50:  6.40E+3nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037844((S)-1-[(S)-3-({(2R,4S)-2-[Benzylcarbamoyl-((S)-phe...)
Affinity DataIC50:  6.50E+3nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037823((2R,4S)-2-[Benzylcarbamoyl-((S)-phenylacetylamino)...)
Affinity DataIC50: >3.50E+4nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Research And Development

Curated by ChEMBL
LigandPNGBDBM50037838((2R,4S)-2-[Benzylcarbamoyl-((S)-phenylacetylamino)...)
Affinity DataIC50: >3.50E+4nMAssay Description:In vitro inhibitory activity against HIV proteinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed