Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50036294
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368919(CHEMBL608026)
Affinity DataKi:  74nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118811(5-(1,3-Dibutyl-2,6-dioxo-1,2,3,6-tetrahydro-purin-...)
Affinity DataKi:  229nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368918(CHEMBL610956)
Affinity DataKi:  602nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368911(CHEMBL608956)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368910(CHEMBL610700)
Affinity DataKi:  1.72E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368913(CHEMBL608945)
Affinity DataKi:  2.19E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368911(CHEMBL608956)
Affinity DataKi:  2.25E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368909(CHEMBL607784)
Affinity DataKi:  2.63E+3nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368917(CHEMBL610675)
Affinity DataKi:  2.70E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368914(CHEMBL608657)
Affinity DataKi:  3.06E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368916(CHEMBL608647)
Affinity DataKi:  3.23E+3nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368916(CHEMBL608647)
Affinity DataKi:  3.72E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368908(CHEMBL610417)
Affinity DataKi:  4.19E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368911(CHEMBL608956)
Affinity DataKi:  4.25E+3nMAssay Description:Displacement of specific [3H]- CGS-21680 in rat striatal membranes A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368910(CHEMBL610700)
Affinity DataKi:  4.51E+3nMAssay Description:Displacement of specific [3H]- CGS-21680 in rat striatal membranes A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368920(CHEMBL610095)
Affinity DataKi:  4.81E+3nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368908(CHEMBL610417)
Affinity DataKi:  6.03E+3nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368918(CHEMBL610956)
Affinity DataKi:  6.21E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368913(CHEMBL608945)
Affinity DataKi:  8.67E+3nMAssay Description:Displacement of specific [3H]- CGS-21680 in rat striatal membranes A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368920(CHEMBL610095)
Affinity DataKi:  8.79E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368915(CHEMBL610372)
Affinity DataKi:  9.10E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368907(CHEMBL611863)
Affinity DataKi:  9.75E+3nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368912(CHEMBL610662)
Affinity DataKi:  1.03E+4nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368909(CHEMBL607784)
Affinity DataKi:  1.12E+4nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368910(CHEMBL610700)
Affinity DataKi:  1.24E+4nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368913(CHEMBL608945)
Affinity DataKi:  1.29E+4nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368914(CHEMBL608657)
Affinity DataKi:  1.53E+4nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368921(CHEMBL610702)
Affinity DataKi:  1.59E+4nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368908(CHEMBL610417)
Affinity DataKi:  1.95E+4nMAssay Description:Displacement of specific [3H]- CGS-21680 in rat striatal membranes A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368912(CHEMBL610662)
Affinity DataKi:  3.08E+4nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118811(5-(1,3-Dibutyl-2,6-dioxo-1,2,3,6-tetrahydro-purin-...)
Affinity DataKi:  3.73E+4nMAssay Description:Tested for the displacement of specific [3H]PIA in rat brain membranes of A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368918(CHEMBL610956)
Affinity DataKi:  3.81E+4nMAssay Description:Displacement of specific [3H]- CGS-21680 in rat striatal membranes A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368907(CHEMBL611863)
Affinity DataKi:  4.30E+4nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368920(CHEMBL610095)
Affinity DataKi:  4.73E+4nMAssay Description:Displacement of specific [3H]- CGS-21680 in rat striatal membranes A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368915(CHEMBL610372)
Affinity DataKi:  5.35E+4nMAssay Description:Displacement of specific [3H]- CGS-21680 in rat striatal membranes A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368914(CHEMBL608657)
Affinity DataKi:  5.49E+4nMAssay Description:Displacement of specific [3H]- CGS-21680 in rat striatal membranes A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368921(CHEMBL610702)
Affinity DataKi:  8.12E+4nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368917(CHEMBL610675)
Affinity DataKi:  8.94E+4nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368915(CHEMBL610372)
Affinity DataKi:  2.28E+5nMAssay Description:Displacement of specific [125]AB-MECA binding in membranes of CHO cells stably transfected with the rat A3-cDNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed