Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50036314
LigandPNGBDBM50040692((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propyl...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory activity against bovine type-1 geranylgeranyl transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040692((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propyl...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040690((S)-2-{(S)-2-[(S)-2-(2-Amino-3-mercapto-propylamin...)
Affinity DataIC50:  4.80nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040689((S)-2-{(S)-2-[(S)-2-(2-Amino-3-mercapto-propylamin...)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040689((S)-2-{(S)-2-[(S)-2-(2-Amino-3-mercapto-propylamin...)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity against bovine type-1 geranylgeranyl transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50407296(CHEMBL2052018 | L-731735)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040691((S)-2-{(S)-2-[(S)-2-(2-Amino-3-mercapto-propionyla...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040691((S)-2-{(S)-2-[(S)-2-(2-Amino-3-mercapto-propionyla...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against bovine type-1 geranylgeranyl transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040684((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propyl...)
Affinity DataIC50:  28nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040684((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propyl...)
Affinity DataIC50:  28nMAssay Description:Inhibitory activity against bovine type-1 geranylgeranyl transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040688((S)-2-{(S)-2-[(S)-2-(3-Mercapto-propylamino)-3-met...)
Affinity DataIC50:  29nMAssay Description:Inhibitory activity against bovine type-1 geranylgeranyl transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040688((S)-2-{(S)-2-[(S)-2-(3-Mercapto-propylamino)-3-met...)
Affinity DataIC50:  29nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040683((S)-2-{(S)-2-[(S)-2-(3-Mercapto-propylamino)-3-met...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040685((S)-2-{(S)-2-[(S)-2-(2-Amino-3-mercapto-propylamin...)
Affinity DataIC50:  140nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040695((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propio...)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108076((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propio...)
Affinity DataIC50:  165nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040682((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propio...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040693((S)-2-{(S)-2-[(S)-2-(3-Mercapto-propylamino)-3-met...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040685((S)-2-{(S)-2-[(S)-2-(2-Amino-3-mercapto-propylamin...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro inhibition of bovine type-1 geranylgeranyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040690((S)-2-{(S)-2-[(S)-2-(2-Amino-3-mercapto-propylamin...)
Affinity DataIC50:  5.75E+3nMAssay Description:In vitro inhibition of bovine type-1 geranylgeranyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040694((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propyl...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040694((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propyl...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against bovine type-1 geranylgeranyl transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040693((S)-2-{(S)-2-[(S)-2-(3-Mercapto-propylamino)-3-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of bovine type-1 geranylgeranyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040683((S)-2-{(S)-2-[(S)-2-(3-Mercapto-propylamino)-3-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against bovine type-1 geranylgeranyl transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040687((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propio...)
Affinity DataIC50:  1.13E+4nMAssay Description:Inhibitory activity against bovine type-1 geranylgeranyl transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50040687((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propio...)
Affinity DataIC50:  1.13E+4nMAssay Description:Inhibitory activity against Ras Farnesyl Protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50407296(CHEMBL2052018 | L-731735)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibitory activity against bovine type-1 geranylgeranyl transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50108076((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propio...)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibitory activity against bovine type-1 geranylgeranyl transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed