Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 4928
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50002369((2S-(2alpha,3beta,4beta))-2-carboxy-4-(1-methyleth...)
Affinity DataKi:  2.29nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM17660((2S)-2-amino-3-(3,5-dioxo-1,2,4-oxadiazolidin-2-yl...)
Affinity DataKi:  6.43nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50252103((2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-MET...)
Affinity DataKi:  10.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50013055(2-aminopentanedioateglutamate | L-Glutamate | glut...)
Affinity DataKi:  18.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50002370((R,S)-alpha-amino-3-hydroxy-5-methyl-4-isooxazole-...)
Affinity DataKi:  1.97E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50240399((2R,3R,4S)-3-(carboxymethyl)-4-isopropylpyrrolidin...)
Affinity DataKi:  3.84E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM82560(CAS_2379-57-9 | DNQX | NSC_3140)
Affinity DataKi:  8.49E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50289504(7-Cyano-3-hydroxy-6-nitro-quinoxalin-2-ol anion | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50002343(2-Methylamino-succinic acid | CHEMBL275325 | NMDA)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed